SCHEMBL9734744

SCHEMBL9734744

O=C1CCN(C(=O)Cc2ccc(Cl)c(Cl)c2)C(CN2CCCC2)C1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
OPRK1 P41145 18/20 1.00
NPC1 O15118 1/20 0.72
CYP1A2 P05177 1/20 0.72
CYP3A4 P08684 1/20 0.72
CYP2D6 P10635 1/20 0.72
CYP2C9 P11712 1/20 0.72
NFKB1 P19838 1/20 0.72
CYP2C19 P33261 1/20 0.72
OPRD1 P41143 1/20 0.72
HIF1A Q16665 1/20 0.72
TDP1 Q9NUW8 1/20 0.72
BLM P54132 1/20 0.71
PMP22 Q01453 1/20 0.71
DRD4 P21917 1/20 0.71
SLC6A3 Q01959 1/20 0.71
TMEM97 Q5BJF2 1/20 0.71
SIGMAR1 Q99720 1/20 0.71

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9735327 0.99 OPRK1 (0.98) OPRK1NPC1CYP1A2CYP3A4CYP2D6
SCHEMBL10338867 0.84 OPRK1 (1.00) OPRK1NPC1CYP1A2CYP3A4CYP2D6
SCHEMBL6622624 0.84 OPRK1 (1.00) OPRK1NPC1CYP1A2CYP3A4CYP2D6
Hydrochloric Acid SCHEMBL9734087 0.83 OPRK1 (0.71) OPRK1NPC1CYP1A2CYP3A4CYP2D6
Hydrochloric Acid SCHEMBL9734090 0.83 OPRK1 (0.71) OPRK1NPC1CYP1A2CYP3A4CYP2D6
Hydrochloric Acid SCHEMBL9730605 0.83 OPRK1 (0.95) OPRK1NPC1CYP1A2CYP3A4CYP2D6
Hydrochloric Acid SCHEMBL8435659 0.83 OPRK1 (1.00) OPRK1NPC1CYP1A2CYP3A4CYP2D6
Hydrochloric Acid SCHEMBL7642844 0.83 OPRK1 (1.00) OPRK1NPC1CYP1A2CYP3A4CYP2D6
Hydrochloric Acid SCHEMBL9734221 0.83 OPRK1 (0.98) OPRK1NPC1CYP1A2CYP3A4CYP2D6
Hydrochloric Acid SCHEMBL9731858 0.82 OPRK1 (0.98) OPRK1NPC1CYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5114945-A Spiropiperidine derivatives GLAXO GROUP LIMITED (GB) 1992-05-19 US disclosed