SCHEMBL9735921

SCHEMBL9735921

COc1ccc(CCCCN(C)CC[C@]2(O)CCc3cc(F)ccc3[C@H]2C(C)C)cc1OC

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 11/20 0.58
CYP2D6 P10635 10/20 0.50
CACNA1H O95180 4/20 0.44
MAPT P10636 4/20 0.44
CACNA1B Q00975 3/20 0.44
KCNH2 Q12809 2/20 0.44
CACNA1C Q13936 2/20 0.44
ABCB11 O95342 2/20 0.44
CYP1A2 P05177 2/20 0.44
ABCB1 P08183 2/20 0.44
NPC1 O15118 1/20 0.44
CACNA1G O43497 1/20 0.44
CACNA1F O60840 1/20 0.44
TP53 P04637 1/20 0.44
CHRM2 P08172 1/20 0.44
HTR1A P08908 1/20 0.44
ADRA2A P08913 1/20 0.44
ADORA3 P0DMS8 1/20 0.44
CHRM1 P11229 1/20 0.44
CYP2C9 P11712 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10447243 1.00 CYP3A4 (0.58) CYP3A4CYP2D6CACNA1HMAPTCACNA1B
SCHEMBL10446897 0.97 CYP3A4 (0.61) CYP3A4CYP2D6CACNA1HMAPTCACNA1B
SCHEMBL9736518 0.97 CYP3A4 (0.61) CYP3A4CYP2D6CACNA1HMAPTCACNA1B
SCHEMBL9827446 0.94 CYP3A4 (0.56) CYP3A4CYP2D6CACNA1HMAPTCACNA1B
SCHEMBL9736708 0.94 CYP3A4 (0.56) CYP3A4CYP2D6CACNA1HMAPTCACNA1B
Hydrochloric Acid SCHEMBL9829230 0.93 CYP3A4 (0.55) CYP3A4CYP2D6CACNA1HMAPTCACNA1B
Hydrochloric Acid SCHEMBL9736375 0.93 CYP3A4 (0.55) CYP3A4CYP2D6CACNA1HMAPTCACNA1B
SCHEMBL9829660 0.90 CYP3A4 (0.46) CYP3A4CYP2D6MAPTKCNH2CACNA1C
SCHEMBL9829663 0.90 CYP3A4 (0.46) CYP3A4CYP2D6MAPTKCNH2CACNA1C
Hydrochloric Acid SCHEMBL10792651 0.89 CYP3A4 (0.45) CYP3A4CYP2D6MAPTKCNH2CACNA1C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5120759-A TETRAHYDRONAPHTHALENE DERIVATIVES FOR IMPROVING SHORT-TERM MEMORY HOFFMANN-LA ROCHE INC. (US) 1992-06-09 US disclosed
EP-0388739-A1 Tetrahydronaphthalene derivates F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1990-09-26 EP disclosed