SCHEMBL9736004

SCHEMBL9736004

CSc1ccc(Cn2c(CCC(=O)O)c(C)c3cc(F)ccc32)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGES2 Q9H7Z7 3/20 0.56
HSD17B10 Q99714 2/20 0.56
KDM4E B2RXH2 2/20 0.56
CYP1A2 P05177 2/20 0.56
CYP3A4 P08684 2/20 0.56
CYP2C9 P11712 2/20 0.56
TSHR P16473 2/20 0.56
CYP2C19 P33261 2/20 0.56
MAPT P10636 1/20 0.56
HPGD P15428 1/20 0.56
HIF1A Q16665 1/20 0.56
TDP1 Q9NUW8 1/20 0.56
TBXA2R P21731 2/20 0.48
PTGDR2 Q9Y5Y4 6/20 0.44
AKR1B1 P15121 1/20 0.44
TBXAS1 P24557 2/20 0.43
ALDH1A1 P00352 1/20 0.42
AKR1C3 P42330 1/20 0.41
AKR1C2 P52895 1/20 0.41
LMNA P02545 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9736499 0.88 PTGES2 (0.71) PTGES2HSD17B10KDM4ECYP1A2CYP3A4
SCHEMBL10921726 0.87 PTGES2 (0.58) PTGES2HSD17B10KDM4ECYP1A2CYP3A4
SCHEMBL10510621 0.87 MAPT (0.53) PTGES2HSD17B10KDM4ECYP1A2CYP3A4
SCHEMBL9738239 0.85 AR (0.55) KDM4ECYP1A2CYP3A4CYP2C9TSHR
SCHEMBL10510723 0.84 PTGES2 (0.55) PTGES2HSD17B10KDM4ECYP1A2CYP3A4
SCHEMBL9736106 0.82 PTGES2 (0.69) PTGES2HSD17B10KDM4ECYP1A2CYP3A4
SCHEMBL9452875 0.81 TBXAS1 (0.60) PTGES2HSD17B10KDM4ECYP1A2CYP3A4
SCHEMBL9669694 0.81 MAPT (0.56) PTGES2HSD17B10KDM4ECYP1A2CYP3A4
SCHEMBL9736408 0.80 AR (0.48) KDM4ECYP1A2CYP3A4CYP2C9TSHR
SCHEMBL9452850 0.79 TBXAS1 (0.51) PTGES2HSD17B10KDM4ECYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5081145-A Contractile prostaglandin antagonists MERCK FROSST CANADA, INC. (CA) 1992-01-14 US disclosed
EP-0166591-B1 INDOLE-2-ALKANOIC ACIDS AND THEIR USE AS PROSTAGLANDIN ANTAGONISTS MERCK FROSST CANADA INC. (CA) 1989-11-23 EP disclosed
EP-0166591-A2 Indole-2-alkanoic acids and their use as prostaglandin antagonists MERCK FROSST CANADA INC. (CA) 1986-01-02 EP disclosed