SCHEMBL9736115

SCHEMBL9736115

CCOC(=O)c1ccc(Br)c(Br)c1Br

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.55
CA12 O43570 4/20 0.50
CA1 P00915 4/20 0.50
CA2 P00918 4/20 0.50
CA7 P43166 4/20 0.50
CA9 Q16790 4/20 0.50
CA14 Q9ULX7 4/20 0.50
ALDH1A1 P00352 3/20 0.47
HSD17B10 Q99714 1/20 0.47
KDM4E B2RXH2 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
RXFP1 Q9HBX9 1/20 0.44
CYP4F2 P78329 1/20 0.44
CYP4A11 Q02928 1/20 0.44
ESR1 P03372 1/20 0.43
ESR2 Q92731 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.42
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
CYP1A2 P05177 3/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL292394 0.92 TSHR (0.63) TSHRCA12CA1CA2CA7
SCHEMBL6160953 0.87 TSHR (0.53) TSHRCA12CA1CA2CA7
SCHEMBL7559624 0.86 MAPT (0.51) TSHRCA12CA1CA2CA7
SCHEMBL2903968 0.86 TSHR (0.52) TSHRCA12CA1CA2CA7
SCHEMBL29092380 0.85 TSHR (0.55) TSHRCA12CA1CA2CA7
SCHEMBL27993119 0.85 TSHR (0.55) TSHRCA12CA1CA2CA7
SCHEMBL7514034 0.84 ALDH1A1 (0.51) TSHRCA12CA1CA2CA7
SCHEMBL7523025 0.84 TSHR (0.50) TSHRCA12CA1CA2CA7
SCHEMBL8492599 0.83 MAPT (0.52) TSHRCA12CA1CA2CA7
SCHEMBL9119101 0.82 TSHR (0.45) TSHRCA12CA1CA2CA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0365541-B1 PREPARATION OF 5-ACYLAMINO-2,4,6-TRIIODO- OR TRIBROMO-BENZOIC ACID DERIVATIVES BRACCO S.p.A. (IT) 1992-08-12 EP disclosed
US-5066823-A Rearrangement reaction, contrast agent for radiology BRACCO INDUSTRIA CHEMICA S.P.A. (IT) 1991-11-19 US disclosed
EP-0365541-A1 PREPARATION OF 5-ACYLAMINO-2,4,6-TRIIODO- OR TRIBROMO-BENZOIC ACID DERIVATIVES. BRACCO IND CHIMICA SPA (IT) 1990-05-02 EP disclosed
WO-1988009328-A1 PREPARATION OF 5-ACYLAMINO-2,4,6-TRIIODO- OR TRIBROMO-BENZOIC ACID DERIVATIVES BRACCO INDUSTRIA CHIMICA S.P.A. (IT) 1988-12-01 WO disclosed