SCHEMBL9736685

SCHEMBL9736685

Cc1c(C(C)CC(=O)O)n(Cc2ccc(Cl)cc2)c2ccc(O)cc12

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGES2 Q9H7Z7 7/20 0.51
MAPT P10636 4/20 0.47
CYP1A2 P05177 2/20 0.47
CYP3A4 P08684 2/20 0.47
CYP2C9 P11712 2/20 0.47
TSHR P16473 2/20 0.47
CYP2C19 P33261 2/20 0.47
HIF1A Q16665 2/20 0.47
KDM4E B2RXH2 2/20 0.47
HPGD P15428 1/20 0.47
HSD17B10 Q99714 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
PTGES O14684 1/20 0.46
S1PR3 Q99500 1/20 0.46
PKM P14618 3/20 0.44
ALDH1A1 P00352 2/20 0.44
GAA P10253 2/20 0.44
LMNA P02545 2/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9736794 0.88 PTGES2 (0.62) PTGES2MAPTCYP1A2CYP3A4CYP2C9
SCHEMBL9736724 0.86 LMNA (0.61) PTGES2MAPTCYP1A2CYP3A4CYP2C9
SCHEMBL9739002 0.83 PTGES2 (0.54) PTGES2MAPTCYP1A2CYP3A4CYP2C9
SCHEMBL10511522 0.78 PTGES2 (0.56) PTGES2MAPTCYP1A2CYP3A4CYP2C9
SCHEMBL9736297 0.77 PTGES2 (0.54) PTGES2MAPTCYP1A2CYP3A4CYP2C9
SCHEMBL9434490 0.76 PTGES2 (0.78) PTGES2MAPTCYP1A2CYP3A4CYP2C9
SCHEMBL10074903 0.76 S1PR3 (0.54) MAPTKDM4ES1PR3PKMALDH1A1
SCHEMBL9736654 0.75 PTGES2 (0.55) PTGES2MAPTCYP1A2CYP3A4CYP2C9
SCHEMBL6025562 0.74 MAPT (0.73) MAPTCYP1A2CYP3A4CYP2C9TSHR
SCHEMBL9736621 0.74 PTGES2 (0.60) PTGES2MAPTCYP1A2CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0166591-B1 INDOLE-2-ALKANOIC ACIDS AND THEIR USE AS PROSTAGLANDIN ANTAGONISTS MERCK FROSST CANADA INC. (CA) 1989-11-23 EP claimed
EP-0166591-A2 Indole-2-alkanoic acids and their use as prostaglandin antagonists MERCK FROSST CANADA INC. (CA) 1986-01-02 EP claimed
US-5081145-A Contractile prostaglandin antagonists MERCK FROSST CANADA, INC. (CA) 1992-01-14 US disclosed
EP-0166591-B1 INDOLE-2-ALKANOIC ACIDS AND THEIR USE AS PROSTAGLANDIN ANTAGONISTS MERCK FROSST CANADA INC. (CA) 1989-11-23 EP disclosed
EP-0166591-A2 Indole-2-alkanoic acids and their use as prostaglandin antagonists MERCK FROSST CANADA INC. (CA) 1986-01-02 EP disclosed