SCHEMBL9736726

SCHEMBL9736726

Cc1c(C(=O)O)n(Cc2ccc(Cl)cc2)c2ccc(F)cc12

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGES2 Q9H7Z7 5/20 0.67
MAPT P10636 4/20 0.67
CYP3A4 P08684 2/20 0.67
TSHR P16473 2/20 0.67
HSD17B10 Q99714 2/20 0.67
KDM4E B2RXH2 2/20 0.67
CYP1A2 P05177 1/20 0.67
CYP2C9 P11712 1/20 0.67
HPGD P15428 1/20 0.67
CYP2C19 P33261 1/20 0.67
HIF1A Q16665 1/20 0.67
TDP1 Q9NUW8 1/20 0.67
TP53 P04637 1/20 0.53
PTGDR2 Q9Y5Y4 3/20 0.52
MEN1 O00255 2/20 0.52
KMT2A Q03164 2/20 0.52
ALOX15 P16050 1/20 0.52
ALOX12 P18054 1/20 0.52
PPARG P37231 1/20 0.52
RECQL P46063 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7089579 0.87 MAPT (0.57) PTGES2MAPTCYP3A4TSHRHSD17B10
SCHEMBL9739350 0.87 MAPT (0.60) PTGES2MAPTCYP3A4TSHRHSD17B10
SCHEMBL12803744 0.82 ALDH1A1 (0.68) PTGES2MAPTCYP3A4TSHRHSD17B10
SCHEMBL4614551 0.81 MAPT (0.47) PTGES2MAPTCYP3A4TSHRHSD17B10
SCHEMBL9736499 0.81 PTGES2 (0.71) PTGES2MAPTCYP3A4TSHRHSD17B10
SCHEMBL3252820 0.80 PTGES2 (1.00) PTGES2MAPTCYP3A4TSHRHSD17B10
SCHEMBL21465497 0.80 PTGDR2 (0.58) PTGES2MAPTCYP3A4TSHRHSD17B10
SCHEMBL29503039 0.80 PTGES2 (1.00) PTGES2MAPTCYP3A4TSHRHSD17B10
SCHEMBL9736645 0.80 PTGES2 (0.69) PTGES2MAPTCYP3A4TSHRHSD17B10
SCHEMBL21465486 0.79 MEN1 (0.83) PTGES2MAPTCYP3A4TSHRHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5081145-A Contractile prostaglandin antagonists MERCK FROSST CANADA, INC. (CA) 1992-01-14 US disclosed
EP-0166591-B1 INDOLE-2-ALKANOIC ACIDS AND THEIR USE AS PROSTAGLANDIN ANTAGONISTS MERCK FROSST CANADA INC. (CA) 1989-11-23 EP disclosed
EP-0166591-A2 Indole-2-alkanoic acids and their use as prostaglandin antagonists MERCK FROSST CANADA INC. (CA) 1986-01-02 EP disclosed