SCHEMBL9739202

SCHEMBL9739202

Cc1cccc(N2C(=O)/C(=N/O)c3ccccc32)c1C

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 7/20 0.47
MEN1 O00255 4/20 0.47
ATM Q13315 1/20 0.41
MAPT P10636 5/20 0.41
CTDSP1 Q9GZU7 1/20 0.40
NPSR1 Q6W5P4 2/20 0.39
NR1H2 P55055 1/20 0.39
NR1H3 Q13133 1/20 0.39
KDM5A P29375 1/20 0.39
CFTR P13569 1/20 0.39
LMNA P02545 3/20 0.38
ALDH1A1 P00352 2/20 0.38
KDM4E B2RXH2 1/20 0.38
CASP3 P42574 1/20 0.38
CASP6 P55212 1/20 0.38
SENP8 Q96LD8 1/20 0.38
SENP7 Q9BQF6 1/20 0.38
SENP6 Q9GZR1 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
CYP1A2 P05177 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9739203 1.00 KMT2A (0.47) KMT2AMEN1ATMMAPTCTDSP1
SCHEMBL9734396 0.80 CES1 (0.56) KMT2AMEN1MAPTNPSR1NR1H2
SCHEMBL29168855 0.77 KMT2A (0.62) KMT2AMEN1NR1H2NR1H3KDM5A
SCHEMBL30758617 0.77 KMT2A (0.62) KMT2AMEN1NR1H2NR1H3KDM5A
SCHEMBL6322884 0.76 ALDH1A1 (0.61) KMT2AMEN1MAPTCTDSP1NPSR1
SCHEMBL6322887 0.76 ALDH1A1 (0.61) KMT2AMEN1MAPTCTDSP1NPSR1
SCHEMBL13628014 0.76 ALDH1A1 (0.61) KMT2AMEN1MAPTCTDSP1NPSR1
SCHEMBL9734125 0.74 BCL2A1 (0.40) KMT2AMEN1ATMMAPTCTDSP1
SCHEMBL9734120 0.74 BCL2A1 (0.40) KMT2AMEN1ATMMAPTCTDSP1
SCHEMBL5194875 0.73 TTR (0.65) KMT2AMEN1ATMMAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5155110-A Antiinflammatory agents, analgesics, antipyretics WARNER-LAMBERT COMPANY (US) 1992-10-13 US disclosed
EP-0316630-A1 Novel fenamic acid hydroxamate derivatives having cyclooxygenase and 5-lipoxygenase inhibition WARNER-LAMBERT COMPANY (US) 1989-05-24 EP disclosed
WO-1989003818-A1 NOVEL FENAMIC ACID HYDROXAMATE DERIVATIVES HAVING CYCLOOXYGENASE AND 5-LIPOXYGENASE INHIBITION WARNER-LAMBERT COMPANY (US) 1989-05-05 WO disclosed