SCHEMBL9739258

SCHEMBL9739258

COc1cc2c(cc1O)CCN(CC1CCCN(CCc3ccc(OC)c(OC)c3)C1)C(=O)C2

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHCR7 Q9UBM7 3/20 0.57
HCN4 Q9Y3Q4 3/20 0.52
MAPT P10636 1/20 0.52
CYP3A4 P08684 1/20 0.51
ALOX15 P16050 1/20 0.51
GAA P10253 2/20 0.43
SMPD1 P17405 1/20 0.41
TDP1 Q9NUW8 2/20 0.41
POLB P06746 1/20 0.41
RECQL P46063 1/20 0.41
PDE4B Q07343 1/20 0.40
KDM4E B2RXH2 2/20 0.40
SIGMAR1 Q99720 1/20 0.40
MEN1 O00255 1/20 0.40
ALDH1A1 P00352 1/20 0.40
KMT2A Q03164 1/20 0.40
CHRM2 P08172 1/20 0.40
HTR1A P08908 1/20 0.40
SLC6A4 P31645 1/20 0.40
DRD3 P35462 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9740117 0.95 HCN4 (0.49) DHCR7HCN4MAPTCYP3A4ALOX15
Cilobradine SCHEMBL628133 0.95 HCN4 (0.57) DHCR7HCN4MAPTCYP3A4ALOX15
Cilobradine SCHEMBL30169956 0.95 HCN4 (0.57) DHCR7HCN4MAPTCYP3A4ALOX15
Cilobradine SCHEMBL1855245 0.95 HCN4 (0.57) DHCR7HCN4MAPTCYP3A4ALOX15
Hydrochloric Acid SCHEMBL9739978 0.94 CYP3A4 (0.50) DHCR7HCN4MAPTCYP3A4ALOX15
Cilobradine SCHEMBL9518220 0.94 CYP3A4 (0.58) DHCR7HCN4MAPTCYP3A4ALOX15
Cilobradine SCHEMBL2459609 0.94 CYP3A4 (0.58) DHCR7HCN4MAPTCYP3A4ALOX15
Cilobradine SCHEMBL29896706 0.94 CYP3A4 (0.58) DHCR7HCN4MAPTCYP3A4ALOX15
Cilobradine SCHEMBL9740702 0.94 HCN4 (0.56) DHCR7HCN4MAPTCYP3A4ALOX15
Hydrochloric Acid SCHEMBL9739678 0.91 CYP3A4 (0.57) DHCR7HCN4MAPTCYP3A4ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed
EP-0224794-A2 Cyclic amine derivatives, medicines containing these compounds and process for their preparation Dr. Karl Thomae GmbH (DE) 1987-06-10 EP disclosed