SCHEMBL9739721

SCHEMBL9739721

N#Cc1cccc2[nH]c[c]c12

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MAP2K1 Q02750 1/20 0.42
IMPDH2 P12268 1/20 0.40
IMPDH1 P20839 1/20 0.40
MCL1 Q07820 1/20 0.37
DYRK1A Q13627 3/20 0.33
TSHR P16473 1/20 0.33
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
SLC6A4 P31645 1/20 0.31
HTT P42858 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2300723 0.72 IMPDH2 (0.52) MAP2K1IMPDH2IMPDH1MCL1DYRK1A
SCHEMBL7278872 0.69 MCL1 (0.37) MAP2K1IMPDH2IMPDH1MCL1DYRK1A
SCHEMBL27479367 0.68 HTR2C (0.34) SLC6A4
SCHEMBL6009041 0.64 MAP2K1 (0.53) MAP2K1IMPDH2IMPDH1MCL1DYRK1A
SCHEMBL403956 0.64 IMPDH2 (0.57) MAP2K1IMPDH2IMPDH1MCL1DYRK1A
SCHEMBL30309353 0.64 IMPDH2 (0.57) MAP2K1IMPDH2IMPDH1MCL1DYRK1A
SCHEMBL645878 0.64 CA1 (0.41) MAP2K1MCL1TSHRKDM4EALDH1A1
SCHEMBL9739950 0.63 IMPDH2 (0.41) MAP2K1IMPDH2IMPDH1MCL1DYRK1A
SCHEMBL7299420 0.63 CA1 (0.40) IMPDH2IMPDH1DYRK1ATSHRKDM4E
SCHEMBL10254 0.61 PARP1 (0.50) MAP2K1IMPDH2IMPDH1MCL1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed