SCHEMBL9740267

SCHEMBL9740267

CC(C1CCCCN1CCc1ccc([N+](=O)[O-])cc1)N1CCc2cc3c(cc2CC1=O)OCO3

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 3/20 0.44
SSTR1 P30872 6/20 0.38
SSTR3 P32745 6/20 0.38
KCNJ1 P48048 5/20 0.37
KCNH2 Q12809 5/20 0.37
MGAM O43451 1/20 0.36
ALDH1A1 P00352 2/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
SIGMAR1 Q99720 1/20 0.36
POLB P06746 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9739389 0.99 HRH3 (0.43) HRH3SSTR1SSTR3KCNJ1KCNH2
SCHEMBL9739293 0.88 ABCG2 (0.46) HRH3KCNJ1KCNH2ALDH1A1MEN1
SCHEMBL9740102 0.88 KCNH2 (0.41) HRH3SSTR3KCNH2ALDH1A1SIGMAR1
Hydrochloric Acid SCHEMBL9740815 0.87 ABCG2 (0.46) HRH3KCNJ1KCNH2ALDH1A1MEN1
SCHEMBL9739283 0.87 HRH3 (0.41) HRH3ALDH1A1MEN1KMT2A
Hydrochloric Acid SCHEMBL9739083 0.86 HRH3 (0.40) HRH3ALDH1A1MEN1KMT2A
SCHEMBL9739319 0.76 SMN1; SMN2 (0.42) HRH3ALDH1A1
Hydrochloric Acid SCHEMBL9740153 0.76 ABCB1 (0.45) HRH3ALDH1A1KMT2A
SCHEMBL9739180 0.76 SMN1; SMN2 (0.43) ALDH1A1
Hydrochloric Acid SCHEMBL9739564 0.76 CYP3A4 (0.41) HRH3ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed
EP-0224794-B1 CYCLIC AMINE DERIVATIVES, MEDICINES CONTAINING THESE COMPOUNDS AND PROCESS FOR THEIR PREPARATION Dr. Karl Thomae GmbH (DE) 1990-09-12 EP disclosed
EP-0224794-A2 Cyclic amine derivatives, medicines containing these compounds and process for their preparation Dr. Karl Thomae GmbH (DE) 1987-06-10 EP disclosed