SCHEMBL9739293

SCHEMBL9739293

COc1cc2c(cc1OC)CC(=O)N(C(C)C1CCCCN1CCc1ccc([N+](=O)[O-])cc1)CC2

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 4/20 0.46
ABCB1 P08183 3/20 0.46
HRH3 Q9Y5N1 3/20 0.45
KCNJ1 P48048 1/20 0.39
KCNH2 Q12809 1/20 0.39
ACHE P22303 2/20 0.39
BCHE P06276 1/20 0.39
MAPT P10636 3/20 0.39
GAA P10253 2/20 0.39
ALDH1A1 P00352 2/20 0.39
KDM4E B2RXH2 1/20 0.39
MEN1 O00255 1/20 0.39
POLB P06746 1/20 0.39
MAPK1 P28482 1/20 0.39
KMT2A Q03164 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
HCN4 Q9Y3Q4 2/20 0.38
LMNA P02545 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9740815 0.99 ABCG2 (0.46) ABCG2ABCB1HRH3KCNJ1KCNH2
SCHEMBL9739319 0.89 SMN1; SMN2 (0.42) ABCG2ABCB1HRH3MAPTGAA
SCHEMBL9740418 0.89 ABCB1 (0.46) ABCG2ABCB1HRH3MAPTGAA
SCHEMBL9739180 0.88 SMN1; SMN2 (0.43) ABCG2ABCB1MAPTGAAALDH1A1
Hydrochloric Acid SCHEMBL9739564 0.88 CYP3A4 (0.41) ABCG2ABCB1HRH3MAPTGAA
Hydrochloric Acid SCHEMBL9740153 0.88 ABCB1 (0.45) ABCG2ABCB1HRH3MAPTGAA
SCHEMBL9740219 0.88 HCN4 (0.49) MAPTGAAALDH1A1KDM4EPOLB
SCHEMBL9739355 0.88 SMN1; SMN2 (0.42) GAAALDH1A1SMN1; SMN2
SCHEMBL9740267 0.88 HRH3 (0.44) HRH3KCNJ1KCNH2ALDH1A1MEN1
SCHEMBL9740525 0.87 HCN4 (0.49) MAPTGAAALDH1A1KDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed
EP-0224794-B1 CYCLIC AMINE DERIVATIVES, MEDICINES CONTAINING THESE COMPOUNDS AND PROCESS FOR THEIR PREPARATION Dr. Karl Thomae GmbH (DE) 1990-09-12 EP disclosed