SCHEMBL9741925

SCHEMBL9741925

BrCCCCCCOCCCCCCc1cnccn1

nearest known ligand 0.31

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.31
HDAC1 Q13547 1/20 0.31
HDAC2 Q92769 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31
HRH1 P35367 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29263707 0.90 HRH1 (0.35) HDAC3HDAC1HDAC2HDAC6HRH1
SCHEMBL31036036 0.90 HRH1 (0.35) HDAC3HDAC1HDAC2HDAC6HRH1
SCHEMBL5159759 0.88 HDAC3 (0.36) HDAC3HDAC1HDAC2HDAC6HRH1
SCHEMBL14835009 0.82 HSP90AA1 (0.34) HDAC3HDAC1HDAC2HDAC6HRH1
SCHEMBL10417000 0.77 HRH1 (0.56) HRH1
SCHEMBL10461495 0.77 HRH1 (0.56) HRH1
SCHEMBL1427937 0.74
SCHEMBL10460727 0.74 HRH1 (0.51) HRH1
SCHEMBL10417735 0.74 HRH1 (0.51) HRH1
SCHEMBL28362525 0.74 HSP90AA1 (0.40) HDAC3HDAC1HDAC2HDAC6HRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5149698-A Pyrimidinyl alkyleneoxy bronchodilator agent GLAXO GROUP LIMITED (GB) 1992-09-22 US disclosed
US-4996218-A Bronchodilator, antiulcer agent, cardiovascular disorders GLAXO GROUP LIMITED (GB) 1991-02-26 US disclosed
EP-0303464-A2 Chloroaniline derivatives GLAXO GROUP LIMITED (GB) 1989-02-15 EP disclosed