SCHEMBL9744094

SCHEMBL9744094

CCOC(=O)C(/C=C(/CP(=O)(OC)OC)C(C)C)NC=O

nearest known ligand 0.34

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.34
CYP3A4 P08684 2/20 0.34
ALOX15 P16050 2/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
TSHR P16473 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
CHRM1 P11229 1/20 0.31
ADORA1 P30542 1/20 0.31
HSD17B10 Q99714 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9743641 0.85 CYP2D6 (0.43) ALDH1A1CYP3A4ALOX15CYP2D6CYP2C9
SCHEMBL9743815 0.84 ALDH1A1 (0.34) ALDH1A1CYP3A4ALOX15CYP2D6CYP2C9
SCHEMBL9742592 0.82 CYP2D6 (0.33) ALDH1A1CYP3A4ALOX15CYP2D6CYP2C9
SCHEMBL9744210 0.82 CYP2D6 (0.33) ALDH1A1CYP3A4ALOX15CYP2D6CYP2C9
SCHEMBL9743713 0.80 CYP2D6 (0.32) ALDH1A1CYP3A4ALOX15CYP2D6CYP2C9
SCHEMBL9743571 0.75 CYP2D6 (0.42) CYP2D6CYP2C9CYP2C19
SCHEMBL9743517 0.75 CYP2D6 (0.42) CYP2D6CYP2C9CYP2C19
SCHEMBL9744920 0.74 CYP2D6 (0.43) CYP2D6CYP2C9CYP2C19TSHR
SCHEMBL8988946 0.73 CYP2D6 (0.30) CYP2D6CYP2C9CYP2C19
SCHEMBL8988987 0.71 CYP2D6 (0.31) CYP2D6CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5175344-A Anticonvulsants, anxiolytic agents CIBA-GEIGY CORPORATION (US) 1992-12-29 US disclosed
EP-0233154-B1 UNSATURATED AMINO-ACIDS CIBA-GEIGY AG (CH) 1991-12-18 EP disclosed
US-5051413-A For treatment of ischemia, antispasmodic agents, anticonvulsants and anxiety or manic conditions CIBA-GEIGY CORPORATION (US) 1991-09-24 US disclosed
EP-0233154-A2 Unsaturated amino-acids CIBA-GEIGY AG (CH) 1987-08-19 EP disclosed