SCHEMBL9745423

SCHEMBL9745423

CC(C)(C)OC(=O)CN(CBr)C(=O)c1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASR P41180 1/20 0.43
ALDH1A1 P00352 3/20 0.43
HPGD P15428 2/20 0.43
CTSS P25774 3/20 0.40
CTSK P43235 1/20 0.40
AKT1 P31749 1/20 0.40
MAPT P10636 1/20 0.40
CTSL P07711 2/20 0.39
CTSB P07858 1/20 0.39
HDAC3 O15379 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC2 Q92769 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
NR1D1 P20393 1/20 0.38
TSHR P16473 1/20 0.38
HSD17B10 Q99714 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
POLB P06746 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2D6 P10635 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27730480 0.87 HPGD (0.55) CASRALDH1A1HPGDMAPTHDAC1
SCHEMBL9743559 0.85 CASR (0.43) CASRALDH1A1HPGDCTSSCTSK
SCHEMBL4182248 0.84 CASR (0.43) CASRALDH1A1HPGDCTSSCTSK
SCHEMBL4177603 0.82 TSHR (0.46) CASRALDH1A1HPGDCTSSCTSK
SCHEMBL9743469 0.77 ALDH1A1 (0.49) ALDH1A1HPGDCTSSMAPTCTSL
SCHEMBL20187564 0.77 AKT1 (0.60) ALDH1A1CTSSAKT1CTSLCTSB
SCHEMBL9540577 0.77 CKS1B (0.49) ALDH1A1HPGDCTSSAKT1CTSL
SCHEMBL4743853 0.74 KMT2A (0.55) CTSSCTSKCTSLCTSBHDAC3
SCHEMBL6437793 0.73 MEN1 (0.42) CASRALDH1A1CTSSAKT1CTSL
SCHEMBL782348 0.73 AKT1 (0.55) CTSSAKT1CTSLCTSBNR1D1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5098996-A Fluorination of compounds for use in diagnosis of nuclear medicine THE UNITED STATES OF AMERICA AS REPRESENTED BY THE DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 1992-03-24 US disclosed