SCHEMBL9747476

SCHEMBL9747476

FC(F)(F)c1cccc(Cn2ccnc2)c1

nearest known ligand 0.72

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 13/20 0.66
CYP11B2 P19099 11/20 0.66
ADRA2C P18825 1/20 0.61
CYP19A1 P11511 6/20 0.58
TBXAS1 P24557 2/20 0.58
CYP1A2 P05177 1/20 0.58
POLB P06746 1/20 0.58
CYP3A4 P08684 1/20 0.58
CYP2D6 P10635 1/20 0.58
MAPT P10636 1/20 0.58
QPCT Q16769 1/20 0.58
CYP4Z1 Q86W10 1/20 0.58
QPCTL Q9NXS2 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11700956 0.85 CYP19A1 (0.64) CYP11B1CYP11B2CYP19A1TBXAS1
SCHEMBL12245400 0.85 CYP11B1 (0.66) CYP11B1CYP11B2ADRA2CCYP19A1TBXAS1
SCHEMBL394308 0.84 CYP11B1 (0.83) CYP11B1CYP11B2ADRA2CCYP19A1TBXAS1
SCHEMBL28140204 0.81 CYP11B1 (0.68) CYP11B1CYP11B2CYP19A1TBXAS1CYP1A2
SCHEMBL9747422 0.80 CYP11B1 (1.00) CYP11B1CYP11B2ADRA2CCYP19A1TBXAS1
SCHEMBL12299569 0.80 CYP11B1 (0.71) CYP11B1CYP11B2ADRA2CCYP19A1TBXAS1
SCHEMBL8070045 0.79 CYP11B1 (0.61) CYP11B1CYP11B2ADRA2CCYP19A1TBXAS1
Hydrochloric Acid SCHEMBL11081394 0.78 EPHX1 (0.46) CYP11B1CYP11B2ADRA2CCYP19A1TBXAS1
SCHEMBL14315492 0.78 CYP11B1 (0.71) CYP11B1CYP11B2CYP19A1TBXAS1CYP1A2
SCHEMBL21950448 0.78 CYP11B1 (0.50) CYP11B1CYP11B2CYP19A1TBXAS1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107922386-A 1,4 disubstituted imidazolium derivatives 大日本住友制药株式会社 2018-04-17 CN disclosed
CN-107922348-A Bicyclic heterocyclic amide derivatives 大日本住友制药株式会社 2018-04-17 CN disclosed
US-5100890-A Antidepressants, Fungicides HOECHST AKTIENGESELLSCHAFT (DE) 1992-03-31 US disclosed
EP-0218118-B1 ARYLMETHYL AZOLES AND THEIR SALTS, METHOD FOR THEIR PREPARATION, COMPOSITIONS CONTAINING THEM AND THEIR USE HOECHST AKTIENGESELLSCHAFT (DE) 1991-09-18 EP disclosed
US-5023357-A Arylmethylazole preparation processes HOECHST AKTIENGESELLSCHAFT (DE) 1991-06-11 US disclosed
US-4876354-A FUNGICIDES, ANTIDEPRESSANTS HOECHST AKTIENGESELLSCHAFT (DE) 1989-10-24 US disclosed
EP-0218118-A1 Arylmethyl azoles and their salts, method for their preparation, compositions containing them and their use HOECHST AKTIENGESELLSCHAFT (DE) 1987-04-15 EP disclosed