SCHEMBL9749159

SCHEMBL9749159

Cn1c(N)cc(=O)n(Cc2ccc(C#N)cc2)c1=O

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 1/20 0.68
CYP3A4 P08684 1/20 0.52
GAA P10253 1/20 0.46
CRHBP P24387 1/20 0.46
CRHR2 Q13324 1/20 0.46
RXFP1 Q9HBX9 1/20 0.46
PARG Q86W56 2/20 0.45
MAPT P10636 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
IDH1 O75874 1/20 0.39
ALDH1A1 P00352 1/20 0.39
P2RX3 P56373 1/20 0.39
KLKB1 P03952 1/20 0.39
KLK1 P06870 1/20 0.39
PIK3R1 P27986 1/20 0.39
PIK3CA P42336 1/20 0.39
CYP19A1 P11511 1/20 0.39
KMT2A Q03164 2/20 0.39
MEN1 O00255 1/20 0.39
CLPP Q16740 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9748739 0.89 CYP3A4 (0.68) HPGDCYP3A4GAACRHBPCRHR2
SCHEMBL28405041 0.79 CYP3A4 (0.47) HPGDCYP3A4GAACRHBPCRHR2
SCHEMBL16028734 0.79 HPGD (0.69) HPGDCYP3A4PARGMAPTALDH1A1
SCHEMBL16845918 0.76 HPGD (0.60) HPGDCYP3A4RXFP1PARGKMT2A
SCHEMBL1944109 0.73 HPGD (0.60) HPGDCYP3A4GAAMAPTALDH1A1
SCHEMBL8443447 0.70 CYP19A1 (0.45) P2RX3CYP19A1HTR2CCA12CA9
SCHEMBL30861151 0.70 CYP19A1 (0.53) HPGDALDH1A1P2RX3CYP19A1HTR2C
SCHEMBL7019248 0.70 MMP13 (0.67) GAACRHBPCRHR2RXFP1PARG
SCHEMBL29142975 0.69 CYP3A4 (1.00) HPGDCYP3A4ALDH1A1KMT2A
SCHEMBL8439059 0.69 CA12 (0.45) MAPTTDP1IDH1ALDH1A1P2RX3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0203721-B1 8-PHENYL XANTHINES THE WELLCOME FOUNDATION LIMITED (GB) 1992-06-10 EP disclosed
US-5017577-A Using Purine Cinnamic Acids BURROUGHS WELLCOME CO. (US) 1991-05-21 US disclosed
US-5015647-A Using Purine Cinnamic Acid Compounds BURROUGHS WELLCOME CO. (US) 1991-05-14 US disclosed
US-4981857-A ADENOSINE ANTAGONIST BURROUGHS WELLCOME CO. (US) 1991-01-01 US disclosed
US-4879296-A BLOCKING ADERNOSINE CELL SURFACE EFFECTS BURROUGHS WELLCOME CO. (US) 1989-11-07 US disclosed
EP-0203721-A2 8-Phenyl xanthines THE WELLCOME FOUNDATION LIMITED (GB) 1986-12-03 EP disclosed