SCHEMBL9749859

SCHEMBL9749859

CNn1cc(C(=O)O)c(=O)c2cc(F)c(N3CCC[C@H]3CO)c(F)c21

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 8/20 0.45
ALDH1A1 P00352 6/20 0.43
HPGD P15428 5/20 0.43
HSD17B10 Q99714 5/20 0.43
PMP22 Q01453 1/20 0.42
LMNA P02545 1/20 0.42
KCNH2 Q12809 3/20 0.40
POLB P06746 2/20 0.39
CHRM2 P08172 1/20 0.39
CHRM1 P11229 1/20 0.39
OPRM1 P35372 1/20 0.39
OPRD1 P41143 1/20 0.39
ALB P02768 1/20 0.39
HRH3 Q9Y5N1 1/20 0.39
ADRA2B P18089 1/20 0.39
MAPK1 P28482 1/20 0.39
TOP2A P11388 1/20 0.39
TOP2B Q02880 1/20 0.39
TOP1 P11387 1/20 0.39
TUBB4A P04350 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10424662 1.00 KDM4E (0.45) KDM4EALDH1A1HPGDHSD17B10PMP22
SCHEMBL9749868 0.88 NTRK1 (0.35) KDM4EALDH1A1HPGDHSD17B10PMP22
SCHEMBL9749882 0.88 KDM4E (0.51) KDM4EALDH1A1HPGDHSD17B10PMP22
SCHEMBL9750386 0.86 KDM4E (0.45) KDM4EALDH1A1HPGDHSD17B10PMP22
SCHEMBL10425104 0.85 TOP2A (0.55) KDM4EALDH1A1HPGDHSD17B10LMNA
SCHEMBL9749871 0.85 TOP2A (0.55) KDM4EALDH1A1HPGDHSD17B10LMNA
SCHEMBL10425075 0.85 KDM4E (0.64) KDM4EALDH1A1HPGDHSD17B10PMP22
SCHEMBL10425078 0.85 KDM4E (0.64) KDM4EALDH1A1HPGDHSD17B10PMP22
SCHEMBL9749297 0.82 KDM4E (0.50) KDM4EALDH1A1HPGDHSD17B10PMP22
SCHEMBL10425974 0.82 KDM4E (0.50) KDM4EALDH1A1HPGDHSD17B10PMP22

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0216345-B1 QUINOLINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1992-02-19 EP disclosed
US-4977265-A WITH BACTERICIDAL ACTIVITY HOFFMANN-LA ROCHE INC. (US) 1990-12-11 US disclosed
US-4946847-A BACTERICIDES HOFFMANN-LA ROCHE INC. (US) 1990-08-07 US disclosed
US-4806541-A ANTIBACTERIAL AGENTS HOFFMANN-LA ROCHE INC. (US) 1989-02-21 US disclosed
EP-0216345-A2 Quinoline derivatives F. HOFFMANN-LA ROCHE AG (CH) 1987-04-01 EP disclosed