SCHEMBL9751584

SCHEMBL9751584

C1=NCCN1Nc1cc2ccccc2s1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.37
CYP2A6 P11509 3/20 0.37
SIGMAR1 Q99720 8/20 0.35
GPR6 P46095 1/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
CHRM2 P08172 1/20 0.35
CHRM4 P08173 1/20 0.35
CHRM5 P08912 1/20 0.35
CHRM1 P11229 1/20 0.35
CHRM3 P20309 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
TSHR P16473 1/20 0.35
CYP2C19 P33261 1/20 0.35
THPO P40225 1/20 0.35
SLC6A3 Q01959 1/20 0.35
ADRB2 P07550 1/20 0.34
HDAC3 O15379 1/20 0.34
HDAC4 P56524 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8582363 0.75 IDO1 (0.49) MEN1KMT2A
SCHEMBL562868 0.72 CYP2A6 (0.39) L3MBTL1CYP2A6SIGMAR1MEN1KMT2A
SCHEMBL6583705 0.70 POLB (0.37) CYP2A6MEN1KMT2ACYP2C19HRH4
SCHEMBL1036360 0.70 LMNA (0.34) SIGMAR1KMT2ACYP3A4CYP2D6CYP2C19
SCHEMBL10978597 0.69 CYP2A6 (0.46) CYP2A6ADRB2ASIC3LOXL2DRD2
SCHEMBL6481877 0.68 CYP2A6 (0.47) CYP2A6SIGMAR1ADRB2HDAC3HDAC4
SCHEMBL7099438 0.68 KDM4E (0.48) MEN1KMT2ANPSR1
SCHEMBL9754305 0.65 CYP2A6 (0.44) CYP2A6SIGMAR1ADRB2HDAC3HDAC4
SCHEMBL6642084 0.65 CYP2A6 (0.44) CYP2A6SIGMAR1ADRB2HDAC3HDAC4
SCHEMBL2494058 0.65 CYP2A6 (0.53) CYP2A6ADRB2HDAC3HDAC4HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0422119-A4 BENZOTHIOPHENE DERIVATIVES USEFUL FOR MODIFYING FEEDING BEHAVIOR AND OBSESSIVE-COMPULSIVE BEHAVIOR 1991-11-13 EP disclosed
EP-0422119-A1 BENZOTHIOPHENE DERIVATIVES USEFUL FOR MODIFYING FEEDING BEHAVIOR AND OBSESSIVE-COMPULSIVE BEHAVIOR NEUREX CORPORATION (US) 1991-04-17 EP disclosed
US-4971974-A ANOREXIGENIC AGENTS, BENZO B!THIENO 2,3-C!PYRIDINE COMPOUNDS NEUREX CORPORATION (US) 1990-11-20 US disclosed
WO-1989012447-A1 BENZOTHIOPHENE DERIVATIVES USEFUL FOR MODIFYING FEEDING BEHAVIOR AND OBSESSIVE-COMPULSIVE BEHAVIOR NEUREX CORPORATION (US) 1989-12-28 WO disclosed