SCHEMBL9752147

SCHEMBL9752147

CC(C)(C)OC(=O)N[C@H]1CCc2ccc(N)cc2C1

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 4/20 0.50
MTNR1B P49286 4/20 0.50
NR1H2 P55055 1/20 0.49
CA1 P00915 4/20 0.47
CA2 P00918 4/20 0.47
ACHE P22303 4/20 0.47
EPHX2 P34913 1/20 0.46
DRD2 P14416 4/20 0.45
CTSK P43235 2/20 0.43
BTK Q06187 1/20 0.43
KDM1A O60341 1/20 0.41
MAOB P27338 1/20 0.41
KCNA3 P22001 1/20 0.41
NFKB1 P19838 1/20 0.41
NFKB2 Q00653 1/20 0.41
RELA Q04206 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9752143 1.00 MTNR1A (0.50) MTNR1AMTNR1BNR1H2CA1CA2
SCHEMBL17478343 0.95 CA1 (0.47) MTNR1AMTNR1BNR1H2CA1CA2
SCHEMBL13263584 0.95 CA1 (0.47) MTNR1AMTNR1BNR1H2CA1CA2
SCHEMBL17478424 0.95 CA1 (0.47) MTNR1AMTNR1BNR1H2CA1CA2
SCHEMBL5598167 0.89 EPHX2 (0.50) NR1H2CA1CA2EPHX2DRD2
SCHEMBL5677299 0.86 CA1 (0.64) MTNR1AMTNR1BCA1CA2ACHE
SCHEMBL5722246 0.86 CA1 (0.64) MTNR1AMTNR1BCA1CA2ACHE
SCHEMBL9136687 0.86 CA1 (0.64) MTNR1AMTNR1BCA1CA2ACHE
SCHEMBL464262 0.85 MTNR1A (0.50) MTNR1AMTNR1BCA1CA2ACHE
SCHEMBL9132121 0.82 MTNR1A (0.48) MTNR1AMTNR1BCA1CA2ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5053430-A For treating schizophrenia BOEHRINGER INGELHEIM KG (DE) 1991-10-01 US disclosed
EP-0435988-A1 2-AMINO-7-CARBAMOYL-1,2,3,4-TETRAHYDRONAPHTHALENES, PROCESS FOR PREPARING THEM AND THEIR USE AS DRUGS BOEHRINGER INGELHEIM KG (DE) 1991-07-10 EP disclosed
WO-1991001297-A1 2-AMINO-7-CARBAMOYL-1,2,3,4-TETRAHYDRONAPHTHALENES, PROCESS FOR PREPARING THEM AND THEIR USE AS DRUGS BOEHRINGER INGELHEIM KG (DE) 1991-02-07 WO disclosed
EP-0361300-A1 Use of 2,7 diamino-1,2,3,4-tetrahydronaphthalenes as drugs, 2,7 diamino-1,2,3,4-tetrahydronaphthalenes as well as processes for their preparation BOEHRINGER INGELHEIM KG (DE) 1990-04-04 EP disclosed