SCHEMBL9753228

SCHEMBL9753228

CC(C)c1c(C=CC=O)c(-c2ccc(F)cc2)nn2c(Cl)ccc12

nearest known ligand 0.39

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 3/20 0.39
PTGS2 P35354 12/20 0.34
PTGS1 P23219 1/20 0.33
KDM5B Q9UGL1 1/20 0.33
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9753226 1.00 MAPK14 (0.39) MAPK14PTGS2PTGS1KDM5BKMT2A
SCHEMBL9753114 0.89 MAPK14 (0.42) MAPK14PTGS2PTGS1KDM5BKMT2A
SCHEMBL9752990 0.88 KDM5B (0.34) MAPK14PTGS2PTGS1KDM5B
SCHEMBL9753686 0.88 MAPK14 (0.40) MAPK14PTGS2PTGS1KDM5BKMT2A
SCHEMBL9752989 0.88 KDM5B (0.34) MAPK14PTGS2PTGS1KDM5B
SCHEMBL9753682 0.88 MAPK14 (0.40) MAPK14PTGS2PTGS1KDM5BKMT2A
SCHEMBL9753463 0.87 PTGS2 (0.34) MAPK14PTGS2PTGS1KDM5B
SCHEMBL9753466 0.87 PTGS2 (0.34) MAPK14PTGS2PTGS1KDM5B
SCHEMBL9753312 0.85 KDM5B (0.32) PTGS2PTGS1KDM5B
SCHEMBL9753389 0.85 KDM5B (0.32) PTGS2PTGS1KDM5B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1991018903-A1 PYRROLOPYRIDAZINE COMPOUNDS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1991-12-12 WO disclosed