SCHEMBL9760910

SCHEMBL9760910

O=c1[nH]c(=O)c2cc(C(c3ccccc3)n3cncn3)ccc2[nH]1

nearest known ligand 0.56

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 16/20 0.56
CYP26A1 O43174 2/20 0.50
CYP3A4 P08684 1/20 0.41
CYP11B1 P15538 1/20 0.41
TSHR P16473 1/20 0.41
CYP11B2 P19099 1/20 0.41
CYP2C19 P33261 1/20 0.41
FNTA P49354 1/20 0.39
FNTB P49356 1/20 0.39
KDM4E B2RXH2 1/20 0.39
CA12 O43570 1/20 0.39
PARP1 P09874 1/20 0.39
CA9 Q16790 1/20 0.39
STS P08842 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10102450 0.77 CYP19A1 (0.53) CYP19A1CYP26A1CYP3A4CYP11B1TSHR
SCHEMBL13292485 0.75 CYP19A1 (1.00) CYP19A1CYP26A1CYP3A4CYP11B1TSHR
SCHEMBL14565226 0.74 CYP19A1 (0.56) CYP19A1CYP26A1CYP3A4CYP11B1TSHR
SCHEMBL10102510 0.74 CYP19A1 (0.49) CYP19A1CYP26A1CYP11B1KDM4E
SCHEMBL9524108 0.72 CYP19A1 (0.60) CYP19A1CYP26A1CYP3A4CYP11B1TSHR
SCHEMBL12337077 0.72 CYP19A1 (0.49) CYP19A1CYP26A1CYP11B1KDM4E
SCHEMBL9761076 0.72 KDM4E (0.50) KDM4ECA12PARP1CA9
SCHEMBL7413890 0.71 CYP19A1 (0.83) CYP19A1CYP26A1CYP3A4CYP11B1TSHR
SCHEMBL9760022 0.70 CYP19A1 (0.56) CYP19A1CYP26A1CYP3A4CYP11B1CYP11B2
SCHEMBL11367077 0.69 CYP19A1 (0.79) CYP19A1CYP26A1CYP3A4CYP11B1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5037829-A Antitumor Activity; Androgen, Estrogen Inhibitors; Suppress The Plasma Elimination Of Retinoids JANSSEN PHARMACEUTICA N.V. (BE) 1991-08-06 US disclosed