SCHEMBL9762771

SCHEMBL9762771

O=C1Cc2cc3c(cc2N1)NCN3

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
AHR P35869 4/20 0.48
CMA1 P23946 2/20 0.48
PDE3B Q13370 2/20 0.47
PDE3A Q14432 2/20 0.47
EIF2AK2 P19525 1/20 0.47
PDK2 Q15119 1/20 0.45
CYP1A2 P05177 1/20 0.41
CYP11B1 P15538 1/20 0.41
CYP11B2 P19099 1/20 0.41
EPHX2 P34913 1/20 0.41
PGR P06401 3/20 0.40
GRIA1 P42261 2/20 0.40
CACNG8 Q8WXS5 2/20 0.40
KIF11 P52732 2/20 0.39
GAA P10253 1/20 0.37
CRBN Q96SW2 1/20 0.37
MAOB P27338 1/20 0.36
CA9 Q16790 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31010750 0.87 AHR (0.59) AHRCMA1PDE3BPDE3AEIF2AK2
SCHEMBL9834566 0.75 AHR (0.44) AHRCMA1PDE3BPDE3AEIF2AK2
SCHEMBL548762 0.72 AHR (0.50) AHRCMA1PDE3BPDE3AEIF2AK2
SCHEMBL1436084 0.72 GRIA1 (0.53) AHRCMA1PDE3BPDE3AEIF2AK2
SCHEMBL5441646 0.72 AHR (0.60) AHRCMA1PDE3BPDE3AEIF2AK2
SCHEMBL4065845 0.72 AHR (0.60) AHRCMA1PDE3BPDE3AEIF2AK2
SCHEMBL9298074 0.72 AHR (0.50) AHRCMA1PDE3BPDE3AEIF2AK2
SCHEMBL2491904 0.72 AHR (0.50) AHRCMA1PDE3BPDE3AEIF2AK2
SCHEMBL578508 0.72 SRC (0.57) AHRCMA1PDE3BPDE3AEIF2AK2
SCHEMBL18388811 0.71 HDAC1 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4981864-A ANTICOAGULANTS BOEHRINGER MANNEHIM GMBH (DE) 1991-01-01 US disclosed