Bromide

Bromide

SCHEMBL9763311

Br.NC(=O)Nc1ccc(CCOCCCCCCNCC(O)c2ccc(O)c(CO)c2)cc1

nearest known ligand 0.76

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 known ✓ P07550 19/20 0.76
ADRB3 known ✓ P13945 19/20 0.76
ADRB1 known ✓ P08588 18/20 0.76
HTR1A known ✓ P08908 1/20 0.67
ADRA2B known ✓ P18089 1/20 0.67
SLC6A2 known ✓ P23975 1/20 0.67
ADRA1D known ✓ P25100 1/20 0.67
HTR1D known ✓ P28221 1/20 0.67
HTR1B known ✓ P28222 1/20 0.67
SLC6A4 known ✓ P31645 1/20 0.67
ADRA1A known ✓ P35348 1/20 0.67
SLC6A3 known ✓ Q01959 1/20 0.67
KDM4E B2RXH2 1/20 0.67
CHRM5 P08912 1/20 0.67
DRD2 P14416 1/20 0.67
DRD4 P21917 1/20 0.67
FPR3 P25089 1/20 0.67
HTR2A P28223 1/20 0.67
HTR2C P28335 1/20 0.67
GPR183 P32249 1/20 0.67

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9763066 0.91 ADRB2 (0.74) ADRB2ADRB3ADRB1KDM4EHTR1A
SCHEMBL9763332 0.90 ADRB2 (0.75) ADRB2ADRB3ADRB1KDM4EHTR1A
SCHEMBL9763363 0.87 ADRB2 (0.71) ADRB2ADRB3ADRB1KDM4EHTR1A
SCHEMBL9762577 0.87 ADRB2 (0.79) ADRB2ADRB3ADRB1KDM4EHTR1A
SCHEMBL9763403 0.86 ADRB2 (0.70) ADRB2ADRB3ADRB1KDM4EHTR1A
SCHEMBL9763108 0.86 ADRB2 (0.73) ADRB2ADRB3ADRB1KDM4EHTR1A
SCHEMBL5471417 0.86 ADRB2 (1.00) ADRB2ADRB3ADRB1KDM4EHTR1A
SCHEMBL5450250 0.86 ADRB2 (1.00) ADRB2ADRB3ADRB1KDM4EHTR1A
SCHEMBL5447178 0.86 ADRB2 (1.00) ADRB2ADRB3ADRB1KDM4EHTR1A
SCHEMBL5450243 0.86 ADRB2 (1.00) ADRB2ADRB3ADRB1KDM4EHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4990505-A Treating asthma, bronchitis; adrenergic stimulants GLAXO GROUP LIMITED (GB) 1991-02-05 US disclosed