SCHEMBL9764064

SCHEMBL9764064

CC(C)n1c(C(=O)O)c(-c2ccc(F)cc2)c2ccccc2c1=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HMGCR P04035 6/20 0.46
CYP2C9 P11712 4/20 0.46
SIRT6 Q8N6T7 2/20 0.46
ABCC3 O15438 1/20 0.46
ABCB11 O95342 1/20 0.46
PGR P06401 1/20 0.46
ADORA3 P0DMS8 1/20 0.46
RXRA P19793 1/20 0.46
TBXA2R P21731 1/20 0.46
CCKAR P32238 1/20 0.46
ADRA1A P35348 1/20 0.46
PTGS2 P35354 1/20 0.46
NR4A2 P43354 1/20 0.46
PDE4D Q08499 1/20 0.46
SLC10A1 Q14973 1/20 0.46
TACR1 P25103 2/20 0.43
KDM4E B2RXH2 3/20 0.42
LMNA P02545 2/20 0.42
ALDH1A1 P00352 2/20 0.42
TDP1 Q9NUW8 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9764097 0.88 TACR1 (0.44) HMGCRCYP2C9SIRT6ABCC3ABCB11
SCHEMBL9441598 0.85 HMGCR (0.57) HMGCRCYP2C9SIRT6ABCC3ABCB11
SCHEMBL8948131 0.82 TACR1 (0.55) TACR1KDM4ELMNAALDH1A1TDP1
SCHEMBL10515169 0.82 CDC25A (0.45) HMGCRCYP2C9SIRT6ABCC3ABCB11
SCHEMBL10515162 0.80 CDC25A (0.43) HMGCRCYP2C9SIRT6ABCC3ABCB11
SCHEMBL9461496 0.79 CYP2C9 (0.52) HMGCRCYP2C9SIRT6ABCC3ABCB11
SCHEMBL9461492 0.79 CYP2C9 (0.52) HMGCRCYP2C9SIRT6ABCC3ABCB11
SCHEMBL9764062 0.79 CDC25A (0.44) HMGCRCYP2C9SIRT6ABCC3ABCB11
SCHEMBL9763495 0.77 CYP2C9 (0.44) HMGCRCYP2C9SIRT6ABCC3ABCB11
SCHEMBL9763589 0.76 MAPK14 (0.43) HMGCRCYP2C9SIRT6ABCC3ABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5004747-A Isoquinolinones MAY & BAKER LIMITED (GB) 1991-04-02 US disclosed
EP-0326386-A2 Isoquinolinones MAY & BAKER LIMITED (GB) 1989-08-02 EP disclosed