SCHEMBL9764062

SCHEMBL9764062

CC(C)n1c(CO)c(-c2ccc(F)cc2)c2ccccc2c1=O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDC25A P30304 1/20 0.44
CDC25C P30307 1/20 0.44
MAPK14 Q16539 2/20 0.43
DPP4 P27487 1/20 0.42
HMGCR P04035 5/20 0.41
CYP2C9 P11712 4/20 0.41
SIRT6 Q8N6T7 2/20 0.41
ABCC3 O15438 1/20 0.41
ABCB11 O95342 1/20 0.41
PGR P06401 1/20 0.41
ADORA3 P0DMS8 1/20 0.41
RXRA P19793 1/20 0.41
TBXA2R P21731 1/20 0.41
CCKAR P32238 1/20 0.41
ADRA1A P35348 1/20 0.41
PTGS2 P35354 1/20 0.41
NR4A2 P43354 1/20 0.41
PDE4D Q08499 1/20 0.41
SLC10A1 Q14973 1/20 0.41
TACR1 P25103 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9763589 0.87 MAPK14 (0.43) CDC25ACDC25CMAPK14DPP4HMGCR
SCHEMBL7141401 0.84 HMGCR (0.50) CDC25ACDC25CMAPK14HMGCRCYP2C9
SCHEMBL10515169 0.82 CDC25A (0.45) CDC25ACDC25CMAPK14HMGCRCYP2C9
Bromide SCHEMBL9763462 0.82 MAPK14 (0.41) CDC25ACDC25CMAPK14DPP4HMGCR
SCHEMBL10515162 0.80 CDC25A (0.43) CDC25ACDC25CMAPK14HMGCRCYP2C9
SCHEMBL9764064 0.79 HMGCR (0.46) HMGCRCYP2C9SIRT6ABCC3ABCB11
SCHEMBL9764097 0.78 TACR1 (0.44) CDC25ACDC25CHMGCRCYP2C9SIRT6
SCHEMBL9763495 0.77 CYP2C9 (0.44) CDC25ACDC25CMAPK14HMGCRCYP2C9
SCHEMBL6091326 0.76 HMGCR (0.68) MAPK14HMGCRCYP2C9SIRT6ABCC3
SCHEMBL5731806 0.75 HMGCR (0.54) HMGCR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5004747-A Isoquinolinones MAY & BAKER LIMITED (GB) 1991-04-02 US disclosed
EP-0326386-A2 Isoquinolinones MAY & BAKER LIMITED (GB) 1989-08-02 EP disclosed