SCHEMBL9764438

SCHEMBL9764438

Cc1cc2c(cc1O)[C@@H](c1ccccc1)CN(C)CC2

nearest known ligand 0.82

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD1 P21728 15/20 0.82
HSD17B10 Q99714 4/20 0.82
THPO P40225 2/20 0.82
MAPK1 P28482 2/20 0.82
HIF1A Q16665 1/20 0.82
MTOR P42345 1/20 0.82
DRD2 P14416 4/20 0.81
KDM4E B2RXH2 1/20 0.81
MAPT P10636 1/20 0.81
BLM P54132 1/20 0.81
PMP22 Q01453 1/20 0.81
SMN1; SMN2 Q16637 1/20 0.81
DRD5 P21918 4/20 0.75
CYP1A2 P05177 3/20 0.75
CYP2D6 P10635 3/20 0.75
TSHR P16473 3/20 0.75
CYP3A4 P08684 1/20 0.75
NFKB1 P19838 1/20 0.75
CYP2C19 P33261 1/20 0.75
ADCY2 Q08462 1/20 0.75

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13928823 0.95 DRD1 (0.82) DRD1HSD17B10THPOMAPK1HIF1A
SCHEMBL11712694 0.91 DRD1 (1.00) DRD1HSD17B10THPOMAPK1HIF1A
Bromide SCHEMBL11707024 0.89 KDM4E (1.00) DRD1HSD17B10THPOMAPK1HIF1A
SCHEMBL16263409 0.89 DRD1 (0.72) DRD1HSD17B10THPOMAPK1HIF1A
Sch-23390 SCHEMBL11107859 0.86 DRD1 (1.00) DRD1HSD17B10THPOMAPK1HIF1A
SCHEMBL11398674 0.86 DRD1 (1.00) DRD1HSD17B10THPOMAPK1HIF1A
SCHEMBL469504 0.86 DRD1 (0.81) DRD1HSD17B10THPOMAPK1HIF1A
Sch-23390 SCHEMBL2916216 0.86 DRD1 (1.00) DRD1HSD17B10THPOMAPK1HIF1A
SCHEMBL31676580 0.86 DRD1 (0.81) DRD1HSD17B10THPOMAPK1HIF1A
Sch-23390 SCHEMBL16187032 0.86 DRD1 (1.00) DRD1HSD17B10THPOMAPK1HIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4996202-A 1,2,4,5 tetrahydro benzazepine-3 compounds and antipsychotic use thereof SCHERING CORPORATION (US) 1991-02-26 US disclosed