SCHEMBL976446

SCHEMBL976446

O=C(NO)c1sc(-c2ccc(N3CCOCC3)cc2)nc1-c1ccccc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDC7 O00311 3/20 0.62
DBF4 Q9UBU7 3/20 0.62
ALDH1A1 P00352 4/20 0.57
GAA P10253 2/20 0.57
HPGD P15428 1/20 0.57
HTT P42858 2/20 0.53
LMNA P02545 2/20 0.53
ALOX5 P09917 2/20 0.52
L3MBTL1 Q9Y468 1/20 0.52
CNR1 P21554 1/20 0.50
HDAC1 Q13547 2/20 0.49
DGAT1 O75907 1/20 0.49
HDAC3 O15379 1/20 0.49
HDAC4 P56524 1/20 0.49
HDAC7 Q8WUI4 1/20 0.49
HDAC2 Q92769 1/20 0.49
HDAC10 Q969S8 1/20 0.49
HDAC11 Q96DB2 1/20 0.49
HDAC8 Q9BY41 1/20 0.49
HDAC6 Q9UBN7 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL975727 0.83 CDC7 (0.86) CDC7DBF4ALDH1A1GAAHPGD
SCHEMBL14148655 0.81 ALDH1A1 (0.56) CDC7DBF4ALDH1A1GAAHPGD
SCHEMBL978412 0.81 NPC1 (0.55) CDC7DBF4ALDH1A1GAAHDAC1
SCHEMBL978378 0.77 CDC7 (1.00) CDC7DBF4ALDH1A1GAAHPGD
SCHEMBL12336010 0.77 CD274 (0.60) HPGDHTTLMNA
SCHEMBL977661 0.76 CDC7 (0.70) CDC7DBF4ALDH1A1HPGDLMNA
SCHEMBL976273 0.74 CDC7 (0.60) CDC7DBF4ALDH1A1HPGDLMNA
SCHEMBL976455 0.74 CDC7 (0.57) CDC7DBF4ALDH1A1HDAC1HDAC3
SCHEMBL15978879 0.73 AR (0.53) ALDH1A1GAAHPGDHTTLMNA
SCHEMBL15978869 0.73 AR (0.56) ALDH1A1GAAHPGDHTTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8673911-B2 Inhibitors of histone deacetylase METHYLGENE INC. (CA) 2014-03-18 US disclosed
US-8673911-B2 Inhibitors of histone deacetylase METHYLGENE INC. (CA) 2014-03-18 US disclosed
US-8673911-B2 Inhibitors of histone deacetylase METHYLGENE INC. (CA) 2014-03-18 US disclosed
US-20140045850-A1 INHIBITORS OF HISTONE DEACETYLASE METHYLGENE INC. (CA) 2014-02-13 US disclosed
US-20140045850-A1 INHIBITORS OF HISTONE DEACETYLASE METHYLGENE INC. (CA) 2014-02-13 US disclosed
US-20140045850-A1 INHIBITORS OF HISTONE DEACETYLASE METHYLGENE INC. (CA) 2014-02-13 US disclosed
US-20110021771-A1 INHIBITORS OF HISTONE DEACETYLASE METHYLGENE INC. (CA) 2011-01-27 US disclosed
US-20110021771-A1 INHIBITORS OF HISTONE DEACETYLASE METHYLGENE INC. (CA) 2011-01-27 US disclosed
US-20110021771-A1 INHIBITORS OF HISTONE DEACETYLASE METHYLGENE INC. (CA) 2011-01-27 US disclosed
EP-2217588-A1 INHIBITORS OF HISTONE DEACETYLASE Methylgene, Inc. (CA) 2010-08-18 EP disclosed
WO-2009055917-A1 INHIBITORS OF HISTONE DEACETYLASE METHYLGENE INC. (CA) 2009-05-07 WO disclosed
WO-2009055917-A1 INHIBITORS OF HISTONE DEACETYLASE METHYLGENE INC. (CA) 2009-05-07 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110021771-A1 INHIBITORS OF HISTONE DEACETYLASE HDAC1, HDAC11, HDAC3 CDC7 2481/4885DBF4 1443/4885ALDH1A1 699/4885
US-20140045850-A1 INHIBITORS OF HISTONE DEACETYLASE HDAC1, HDAC11, HDAC3 CDC7 2481/4885DBF4 1443/4885ALDH1A1 699/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.