SCHEMBL9765699

SCHEMBL9765699

COC(=O)C1=C(C)NC(C)=C(C(=O)OC2CCCC2)C1c1cccc([N+](=O)[O-])c1

nearest known ligand 0.80

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 2/20 0.71
HIF1A Q16665 3/20 0.71
MEN1 O00255 2/20 0.71
CYP1A2 P05177 2/20 0.71
CYP3A4 P08684 2/20 0.71
CYP2C9 P11712 2/20 0.71
CYP2C19 P33261 2/20 0.71
KMT2A Q03164 2/20 0.71
MAPT P10636 2/20 0.71
LMNA P02545 1/20 0.71
POLB P06746 1/20 0.71
MAPK1 P28482 1/20 0.71
GPR55 Q9Y2T6 1/20 0.71
CYP2D6 P10635 1/20 0.71
TSHR P16473 1/20 0.71
NFKB1 P19838 1/20 0.71
THPO P40225 1/20 0.71
NR3C2 P08235 1/20 0.70
ADORA3 P0DMS8 2/20 0.68
CACNA1C Q13936 2/20 0.68

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9765742 0.92 ABCB1 (0.64) ABCB1HIF1AMEN1CYP1A2CYP3A4
SCHEMBL10746880 0.91 ABCB1 (0.63) ABCB1HIF1AMEN1CYP1A2CYP3A4
SCHEMBL10911103 0.91 ABCB1 (0.65) ABCB1HIF1AMEN1CYP1A2CYP3A4
SCHEMBL11012196 0.90 CACNA1C (0.61) ABCB1HIF1AMEN1CYP1A2CYP3A4
Hydrochloric Acid SCHEMBL7270464 0.90 ABCB1 (0.64) ABCB1HIF1AMEN1CYP1A2CYP3A4
SCHEMBL6455299 0.89 HIF1A (0.87) ABCB1HIF1AMEN1CYP1A2CYP3A4
SCHEMBL30648615 0.89 HIF1A (0.87) ABCB1HIF1AMEN1CYP1A2CYP3A4
SCHEMBL11063168 0.89 CACNA1F (0.79) ABCB1HIF1AMEN1CYP1A2CYP3A4
Hydrochloric Acid SCHEMBL10464260 0.88 HIF1A (0.85) ABCB1HIF1AMEN1CYP1A2CYP3A4
Hydrochloric Acid SCHEMBL4661064 0.88 HIF1A (0.85) ABCB1HIF1AMEN1CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4988717-A Optically active 1,4-dihydropyridine esters useful for treating circulatory illnesses BAYER AKTIENGESELLSCHAFT (DE) 1991-01-29 US disclosed
US-4849433-A The compound, (⃡)1,4-dihydro-2,6-dimethyl-4-(2'-nitrophenyl)-pyridine-3,5-dicarboxylic acid, methyl isobutyl ester, compositions containing same and a method for effecting coronary dilation BAYER AKTIENGESELLSCHAFT (DE) 1989-07-18 US disclosed
US-4703119-A Intermediates of optically active 1,4-dihydropyridines BAYER AKTIENGESELLSCHAFT (DE) 1987-10-27 US disclosed
US-4510310-A 1,4-Dihydro-2,6-dimethyl-4-(2'-chlorophenyl)-3,5-dicarboxylic acid,methyl or ethyl,trifluoroethyl ester BAYER AKTIENGESELLSCHAFT (DE) 1985-04-09 US disclosed