SCHEMBL9765742

SCHEMBL9765742

CC1=C(C(=O)O)C(c2cccc([N+](=O)[O-])c2)C(C(=O)OC2CCCC2)=C(C)N1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 2/20 0.64
CACNA1C Q13936 5/20 0.64
CACNA1F O60840 4/20 0.64
CACNA1D Q01668 4/20 0.64
CACNA1S Q13698 4/20 0.64
ADORA3 P0DMS8 2/20 0.64
CACNA1B Q00975 1/20 0.62
PDE1C Q14123 1/20 0.61
PGR P06401 1/20 0.61
CHRM2 P08172 1/20 0.61
HTR1A P08908 1/20 0.61
ADRA2A P08913 1/20 0.61
CHRM1 P11229 1/20 0.61
DRD1 P21728 1/20 0.61
TBXA2R P21731 1/20 0.61
SLC6A2 P23975 1/20 0.61
SLC6A4 P31645 1/20 0.61
ADRA1A P35348 1/20 0.61
OPRM1 P35372 1/20 0.61
DRD3 P35462 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10746880 0.99 ABCB1 (0.63) ABCB1CACNA1CCACNA1FCACNA1DCACNA1S
SCHEMBL9765699 0.92 ABCB1 (0.71) ABCB1CACNA1CCACNA1FCACNA1DCACNA1S
SCHEMBL11012196 0.90 CACNA1C (0.61) ABCB1CACNA1CCACNA1FCACNA1DCACNA1S
SCHEMBL11063168 0.89 CACNA1F (0.79) ABCB1CACNA1CCACNA1FCACNA1DCACNA1S
SCHEMBL10750936 0.88 CACNA1F (0.69) CACNA1CCACNA1FCACNA1DCACNA1SADORA3
SCHEMBL10748113 0.87 CACNA1F (0.68) ABCB1CACNA1CCACNA1FCACNA1DCACNA1S
SCHEMBL10823915 0.87 CACNA1F (0.68) CACNA1CCACNA1FCACNA1DCACNA1SADORA3
SCHEMBL8301434 0.87 CACNA1C (0.57) ABCB1CACNA1CCACNA1FCACNA1DCACNA1S
SCHEMBL9765707 0.86 CACNA1C (0.64) ABCB1CACNA1CCACNA1FCACNA1DCACNA1S
SCHEMBL10823995 0.86 CACNA1C (0.69) CACNA1CCACNA1FCACNA1DCACNA1SADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4988717-A Optically active 1,4-dihydropyridine esters useful for treating circulatory illnesses BAYER AKTIENGESELLSCHAFT (DE) 1991-01-29 US disclosed
US-4849433-A The compound, (⃡)1,4-dihydro-2,6-dimethyl-4-(2'-nitrophenyl)-pyridine-3,5-dicarboxylic acid, methyl isobutyl ester, compositions containing same and a method for effecting coronary dilation BAYER AKTIENGESELLSCHAFT (DE) 1989-07-18 US disclosed
US-4510310-A 1,4-Dihydro-2,6-dimethyl-4-(2'-chlorophenyl)-3,5-dicarboxylic acid,methyl or ethyl,trifluoroethyl ester BAYER AKTIENGESELLSCHAFT (DE) 1985-04-09 US disclosed