SCHEMBL9765753

SCHEMBL9765753

CCOC(=O)C1=C(C)NC(C)=C(C(=O)O)C1c1cccnc1SC

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.56
HSD17B10 Q99714 3/20 0.56
CASP1 P29466 1/20 0.56
CACNA1C Q13936 2/20 0.53
ALDH1A1 P00352 3/20 0.50
CYP2C9 P11712 3/20 0.48
MEN1 O00255 2/20 0.48
CYP1A2 P05177 2/20 0.48
CYP3A4 P08684 2/20 0.48
CYP2C19 P33261 2/20 0.48
KMT2A Q03164 2/20 0.48
HIF1A Q16665 2/20 0.48
ADORA3 P0DMS8 2/20 0.48
GAA P10253 2/20 0.48
TSHR P16473 2/20 0.48
HPGD P15428 1/20 0.48
TP53 P04637 1/20 0.48
CYP2D6 P10635 1/20 0.48
NFKB1 P19838 1/20 0.48
THPO P40225 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Mesudipine SCHEMBL1900480 0.95 KDM4E (0.60) KDM4EHSD17B10CASP1CACNA1CALDH1A1
SCHEMBL9765777 0.91 KDM4E (0.59) KDM4EHSD17B10CASP1CACNA1CALDH1A1
SCHEMBL7430107 0.87 KDM4E (0.51) KDM4EHSD17B10CASP1CACNA1CALDH1A1
SCHEMBL11364576 0.78 KDM4E (0.41) KDM4EHSD17B10CASP1CACNA1CALDH1A1
SCHEMBL7266705 0.78 KDM4E (0.90) KDM4EHSD17B10CASP1CACNA1CALDH1A1
SCHEMBL9765762 0.77 KDM4E (0.68) KDM4EHSD17B10CASP1CACNA1CALDH1A1
SCHEMBL10555153 0.77 KDM4E (0.64) KDM4EHSD17B10CASP1CACNA1CALDH1A1
SCHEMBL7273568 0.76 CYP2C9 (0.67) KDM4EHSD17B10CASP1CACNA1CALDH1A1
SCHEMBL11356558 0.76 KDM4E (0.41) KDM4EHSD17B10CASP1CACNA1CALDH1A1
SCHEMBL9833019 0.76 CACNA1C (0.64) KDM4EHSD17B10CASP1CACNA1CALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4988717-A Optically active 1,4-dihydropyridine esters useful for treating circulatory illnesses BAYER AKTIENGESELLSCHAFT (DE) 1991-01-29 US disclosed
US-4849433-A The compound, (⃡)1,4-dihydro-2,6-dimethyl-4-(2'-nitrophenyl)-pyridine-3,5-dicarboxylic acid, methyl isobutyl ester, compositions containing same and a method for effecting coronary dilation BAYER AKTIENGESELLSCHAFT (DE) 1989-07-18 US disclosed
US-4510310-A 1,4-Dihydro-2,6-dimethyl-4-(2'-chlorophenyl)-3,5-dicarboxylic acid,methyl or ethyl,trifluoroethyl ester BAYER AKTIENGESELLSCHAFT (DE) 1985-04-09 US disclosed