SCHEMBL9765762

SCHEMBL9765762

CCOC(=O)C1=C(C)NC(C)=C(C(=O)OC)C1c1cccnc1Cl

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.68
HSD17B10 Q99714 4/20 0.68
CYP2C9 P11712 3/20 0.68
ADORA3 P0DMS8 3/20 0.68
ABCB11 O95342 3/20 0.68
TBXA2R P21731 3/20 0.68
ADRA1A P35348 3/20 0.68
SLC6A3 Q01959 3/20 0.68
MEN1 O00255 2/20 0.68
CYP1A2 P05177 2/20 0.68
CYP3A4 P08684 2/20 0.68
CYP2C19 P33261 2/20 0.68
KMT2A Q03164 2/20 0.68
HIF1A Q16665 2/20 0.68
ABCB1 P08183 2/20 0.68
ADRB3 P13945 2/20 0.68
OPRK1 P41145 2/20 0.68
SCN5A Q14524 2/20 0.68
GAA P10253 2/20 0.68
ALDH1A1 P00352 1/20 0.68

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10555153 0.88 KDM4E (0.64) KDM4EHSD17B10CYP2C9ADORA3ABCB11
SCHEMBL9765711 0.88 KDM4E (0.55) KDM4EHSD17B10CYP2C9ADORA3ABCB11
SCHEMBL10552935 0.87 KDM4E (0.63) KDM4EHSD17B10CYP2C9ADORA3ABCB11
SCHEMBL9765777 0.84 KDM4E (0.59) KDM4EHSD17B10CYP2C9ADORA3ABCB11
SCHEMBL3031020 0.83 ADORA3 (0.82) KDM4EHSD17B10CYP2C9ADORA3ABCB11
Felodipine SCHEMBL8787026 0.81 KDM4E (0.85) KDM4EHSD17B10CYP2C9ADORA3ABCB11
Felodipine SCHEMBL920025 0.81 CYP2C9 (1.00) KDM4EHSD17B10CYP2C9ADORA3ABCB11
SCHEMBL7404689 0.81 CYP2C9 (0.82) KDM4EHSD17B10CYP2C9ADORA3ABCB11
Felodipine SCHEMBL13460298 0.81 CYP2C9 (1.00) KDM4EHSD17B10CYP2C9ADORA3ABCB11
Felodipine SCHEMBL26398 0.81 CYP2C9 (1.00) KDM4EHSD17B10CYP2C9ADORA3ABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4988717-A Optically active 1,4-dihydropyridine esters useful for treating circulatory illnesses BAYER AKTIENGESELLSCHAFT (DE) 1991-01-29 US disclosed
US-4510310-A 1,4-Dihydro-2,6-dimethyl-4-(2'-chlorophenyl)-3,5-dicarboxylic acid,methyl or ethyl,trifluoroethyl ester BAYER AKTIENGESELLSCHAFT (DE) 1985-04-09 US disclosed