SCHEMBL9765799

SCHEMBL9765799

COC(=O)C1=C(C)NC(C)=C(C(=O)OC(C)C#N)C1c1ccccc1Cl

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 6/20 0.54
CYP1A2 P05177 6/20 0.54
CYP3A4 P08684 6/20 0.54
ABCB11 O95342 6/20 0.54
CYP2C19 P33261 5/20 0.54
ADORA3 P0DMS8 5/20 0.54
SCN5A Q14524 5/20 0.54
NR1I2 O75469 5/20 0.54
ALDH1A1 P00352 5/20 0.54
KMT2A Q03164 4/20 0.54
KDM4E B2RXH2 4/20 0.54
HSD17B10 Q99714 4/20 0.54
TBXA2R P21731 4/20 0.54
SLC6A3 Q01959 4/20 0.54
ADRA1A P35348 4/20 0.54
HIF1A Q16665 3/20 0.54
MEN1 O00255 3/20 0.54
OPRK1 P41145 3/20 0.54
CYP2D6 P10635 3/20 0.54
HPGD P15428 3/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3035724 0.86 KDM4E (0.68) CYP2C9CYP1A2CYP3A4ABCB11CYP2C19
SCHEMBL29676073 0.86 KDM4E (0.68) CYP2C9CYP1A2CYP3A4ABCB11CYP2C19
SCHEMBL9765720 0.84 CYP2C9 (0.61) CYP2C9CYP1A2CYP3A4ABCB11CYP2C19
SCHEMBL8297431 0.81 ALDH1A1 (0.58) CYP2C9CYP1A2CYP3A4ABCB11CYP2C19
SCHEMBL15463889 0.81 KDM4E (0.62) CYP2C9CYP1A2CYP3A4ABCB11CYP2C19
SCHEMBL3021914 0.81 KDM4E (0.62) CYP2C9CYP1A2CYP3A4ABCB11CYP2C19
SCHEMBL3026759 0.81 KDM4E (0.62) CYP2C9CYP1A2CYP3A4ABCB11CYP2C19
SCHEMBL7349515 0.81 CYP2C9 (0.52) CYP2C9CYP1A2CYP3A4ABCB11CYP2C19
SCHEMBL11365887 0.81 ALDH1A1 (0.41) CYP2C9CYP1A2CYP3A4ABCB11CYP2C19
SCHEMBL7381112 0.80 KDM4E (0.56) CYP2C9CYP1A2CYP3A4ABCB11CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4988717-A Optically active 1,4-dihydropyridine esters useful for treating circulatory illnesses BAYER AKTIENGESELLSCHAFT (DE) 1991-01-29 US disclosed
US-4849433-A The compound, (⃡)1,4-dihydro-2,6-dimethyl-4-(2'-nitrophenyl)-pyridine-3,5-dicarboxylic acid, methyl isobutyl ester, compositions containing same and a method for effecting coronary dilation BAYER AKTIENGESELLSCHAFT (DE) 1989-07-18 US disclosed
US-4510310-A 1,4-Dihydro-2,6-dimethyl-4-(2'-chlorophenyl)-3,5-dicarboxylic acid,methyl or ethyl,trifluoroethyl ester BAYER AKTIENGESELLSCHAFT (DE) 1985-04-09 US disclosed