SCHEMBL9765877

SCHEMBL9765877

CCCn1c(=O)cc(CN)[nH]c1=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.42
GLA P06280 1/20 0.42
MAPT P10636 1/20 0.42
TSHR P16473 1/20 0.40
PDE4A P27815 6/20 0.39
ADORA2A P29274 6/20 0.39
PDE4B Q07343 6/20 0.39
PDE4C Q08493 6/20 0.39
PDE4D Q08499 6/20 0.39
ADORA2B P29275 4/20 0.39
ADORA3 P0DMS8 3/20 0.39
ADORA1 P30542 3/20 0.39
HPGD P15428 1/20 0.39
BLM P54132 1/20 0.39
PDE3A Q14432 1/20 0.39
HSD17B10 Q99714 1/20 0.39
KDM4E B2RXH2 1/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
ALDH1A1 P00352 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5054519 0.87 SMN1; SMN2 (0.41) SMN1; SMN2GLAMAPTTSHRPDE4A
SCHEMBL1546096 0.79 MAPT (0.49) SMN1; SMN2GLAMAPTTSHRPDE4A
SCHEMBL8355057 0.77 SMN1; SMN2 (0.36) SMN1; SMN2GLAMAPTTSHRPDE4A
SCHEMBL4467734 0.77 TSHR (0.43) SMN1; SMN2GLAMAPTTSHRPDE4A
SCHEMBL10864511 0.76 TSHR (0.39) TSHRPDE4AADORA2APDE4BPDE4C
SCHEMBL10864253 0.76 KMT2A (0.39) SMN1; SMN2GLAMAPTTSHRPDE4A
SCHEMBL3297433 0.75 KMT2A (0.54) SMN1; SMN2GLAMAPTTSHRPDE4A
SCHEMBL9414222 0.75 TSHR (0.52) SMN1; SMN2MAPTTSHRPDE4AADORA2A
SCHEMBL4656127 0.74 MAPT (0.42) MAPTTSHRHSD17B10KDM4EMEN1
SCHEMBL14819960 0.72 TSHR (0.40) SMN1; SMN2GLAMAPTTSHRPDE4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0383868-A4 1,3-UNSYMMETRICAL STRAIGHT CHAIN ALKYL-SUBSTITUTED 8-PHENYLXANTHINES 1991-12-04 EP disclosed
EP-0383868-A1 1,3-UNSYMMETRICAL STRAIGHT CHAIN ALKYL-SUBSTITUTED 8-PHENYLXANTHINES MARION LABORATORIES, INC. (US) 1990-08-29 EP disclosed
WO-1990000056-A1 1,3-UNSYMMETRICAL STRAIGHT CHAIN ALKYL-SUBSTITUTED 8-PHENYLXANTHINES MARION LABORATORIES, INC. (US) 1990-01-11 WO disclosed