SCHEMBL9765879

SCHEMBL9765879

CCCn1c(=O)c2[nH]c(-c3ccccc3)nc2n(C)c1=O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 7/20 0.85
ADORA2A P29274 5/20 0.85
KDM4E B2RXH2 2/20 0.85
CYP1A2 P05177 2/20 0.85
HSD17B10 Q99714 2/20 0.85
MEN1 O00255 1/20 0.85
ALDH1A1 P00352 1/20 0.85
CYP3A4 P08684 1/20 0.85
CYP2C9 P11712 1/20 0.85
CYP2C19 P33261 1/20 0.85
KMT2A Q03164 1/20 0.85
ADORA1 P30542 5/20 0.73
ADORA3 P0DMS8 4/20 0.73
BLM P54132 1/20 0.71
NPSR1 Q6W5P4 1/20 0.71

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL661108 0.92 ADORA2B (1.00) ADORA2BADORA2AKDM4ECYP1A2HSD17B10
SCHEMBL9765873 0.90 ADORA2B (0.70) ADORA2BADORA2AKDM4ECYP1A2HSD17B10
SCHEMBL9765918 0.90 ADORA2B (0.85) ADORA2BADORA2AKDM4ECYP1A2HSD17B10
SCHEMBL7323908 0.84 ADORA2B (0.64) ADORA2BADORA2AKDM4ECYP1A2HSD17B10
SCHEMBL9765909 0.84 ADORA2B (1.00) ADORA2BADORA2AKDM4ECYP1A2HSD17B10
8-Phenyl Theophylline SCHEMBL516432 0.84 ADORA2A (1.00) ADORA2BADORA2AKDM4ECYP1A2HSD17B10
SCHEMBL9840392 0.83 ADORA2B (0.81) ADORA2BADORA2AKDM4ECYP1A2HSD17B10
SCHEMBL1945649 0.83 ADORA2B (1.00) ADORA2BADORA2AADORA1ADORA3
SCHEMBL14564546 0.81 ADORA2B (0.79) ADORA2BADORA2AKDM4ECYP1A2HSD17B10
SCHEMBL24304504 0.80 ADORA2B (0.76) ADORA2BADORA2AKDM4ECYP1A2HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0383868-A4 1,3-UNSYMMETRICAL STRAIGHT CHAIN ALKYL-SUBSTITUTED 8-PHENYLXANTHINES 1991-12-04 EP disclosed
US-5032593-A Anithistamines MARION MERRELL DOW INC. (US) 1991-07-16 US disclosed
EP-0383868-A1 1,3-UNSYMMETRICAL STRAIGHT CHAIN ALKYL-SUBSTITUTED 8-PHENYLXANTHINES MARION LABORATORIES, INC. (US) 1990-08-29 EP disclosed
WO-1990000056-A1 1,3-UNSYMMETRICAL STRAIGHT CHAIN ALKYL-SUBSTITUTED 8-PHENYLXANTHINES MARION LABORATORIES, INC. (US) 1990-01-11 WO disclosed