SCHEMBL9765885

SCHEMBL9765885

CCCn1c(=O)[nH]c(=O)c2[nH]c(-c3ccccc3)nc21

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 12/20 1.00
ADORA2A P29274 8/20 1.00
KDM4E B2RXH2 2/20 0.70
ALDH1A1 P00352 2/20 0.70
CYP1A2 P05177 2/20 0.70
CYP3A4 P08684 2/20 0.70
HSD17B10 Q99714 2/20 0.70
MEN1 O00255 1/20 0.70
CYP2C9 P11712 1/20 0.70
CYP2C19 P33261 1/20 0.70
KMT2A Q03164 1/20 0.70
ADORA1 P30542 4/20 0.61
ADORA3 P0DMS8 4/20 0.61
HPGD P15428 1/20 0.57
TSHR P16473 1/20 0.57
MAPK1 P28482 1/20 0.57
THPO P40225 1/20 0.57
PMP22 Q01453 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7866286 0.88 ADORA2B (0.79) ADORA2BADORA2AKDM4EALDH1A1CYP1A2
SCHEMBL7866612 0.87 ADORA2B (0.77) ADORA2BADORA2AKDM4EALDH1A1CYP1A2
SCHEMBL1946291 0.83 ADORA2B (0.78) ADORA2BADORA2AADORA1ADORA3
SCHEMBL661108 0.83 ADORA2B (1.00) ADORA2BADORA2AKDM4EALDH1A1CYP1A2
SCHEMBL7858226 0.83 ADORA2B (0.70) ADORA2BADORA2AKDM4EALDH1A1CYP1A2
SCHEMBL6889649 0.82 ADORA2B (0.69) ADORA2BADORA2AKDM4EALDH1A1CYP1A2
SCHEMBL3479031 0.81 ADORA2B (0.67) ADORA2BADORA2AKDM4EALDH1A1CYP1A2
SCHEMBL9765918 0.81 ADORA2B (0.85) ADORA2BADORA2AKDM4EALDH1A1CYP1A2
SCHEMBL29494961 0.79 ADORA2B (1.00) ADORA2BADORA2AKDM4EALDH1A1HSD17B10
SCHEMBL7228416 0.78 ADORA2B (0.74) ADORA2BADORA2AKDM4EALDH1A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0383868-A4 1,3-UNSYMMETRICAL STRAIGHT CHAIN ALKYL-SUBSTITUTED 8-PHENYLXANTHINES 1991-12-04 EP disclosed
EP-0383868-A1 1,3-UNSYMMETRICAL STRAIGHT CHAIN ALKYL-SUBSTITUTED 8-PHENYLXANTHINES MARION LABORATORIES, INC. (US) 1990-08-29 EP disclosed
WO-1990000056-A1 1,3-UNSYMMETRICAL STRAIGHT CHAIN ALKYL-SUBSTITUTED 8-PHENYLXANTHINES MARION LABORATORIES, INC. (US) 1990-01-11 WO disclosed