SCHEMBL9767015

SCHEMBL9767015

C=CCOC1=CC(=O)NC1

nearest known ligand 0.51

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.51
PTPRC P08575 1/20 0.36
CA12 O43570 5/20 0.33
CA9 Q16790 5/20 0.33
CA1 P00915 4/20 0.33
POLB P06746 1/20 0.33
PDE4A P27815 1/20 0.33
PDE4B Q07343 1/20 0.33
PDE4C Q08493 1/20 0.33
PDE4D Q08499 1/20 0.33
ADRA2A P08913 1/20 0.32
ADRA2B P18089 1/20 0.32
ADRA2C P18825 1/20 0.32
CA2 P00918 1/20 0.32
CA7 P43166 1/20 0.32
CYP3A4 P08684 1/20 0.30
CYP2A6 P11509 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9767083 0.84 HTT (0.50) HTT
SCHEMBL8665320 0.67 CA9 (0.50) PTPRCCA12CA9CA1CA2
SCHEMBL16425187 0.65 ADRA2A (0.38) PTPRCCA12CA9CA1ADRA2A
SCHEMBL8157783 0.63
SCHEMBL9766990 0.63 HTT (0.43) HTT
SCHEMBL2239455 0.59 PTPRC (0.37) PTPRCCA12CA9CA1POLB
SCHEMBL27974242 0.59 PTPRC (0.46) PTPRCCA12CA9CA1POLB
SCHEMBL8829860 0.59
SCHEMBL13461670 0.58 ADRA2A (0.31) CA12CA9CA1ADRA2AADRA2B
SCHEMBL939327 0.58 PTPRC (0.49) PTPRCCA12CA9CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5072006-A Chemical intermeidate; hypotensive agents, muscle relaxants RECHERCHE SYNTEX FRANCE S.A. (FR) 1991-12-10 US disclosed
US-4997846-A Smooth muscle relaxants, hypotensives RESEARCHE SYNTEX FRANCE, S.A. (FR) 1991-03-05 US disclosed
EP-0377966-A2 Novel benzopyranylpyrrolinone derivatives RECHERCHE SYNTEX FRANCE SA (FR) 1990-07-18 EP disclosed