SCHEMBL9769233

SCHEMBL9769233

CC(=O)c1cccc2nnnn12

nearest known ligand 0.33

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.33
ALDH1A1 P00352 4/20 0.32
TNKS O95271 1/20 0.32
THRB P10828 1/20 0.31
KCNJ1 P48048 4/20 0.31
KDM4E B2RXH2 1/20 0.31
POLB P06746 1/20 0.31
HPGD P15428 1/20 0.31
USP2 O75604 1/20 0.31
GLA P06280 1/20 0.31
MAPT P10636 2/20 0.31
LMNA P02545 1/20 0.30
TP53 P04637 1/20 0.30
GAA P10253 1/20 0.30
EGLN2 Q96KS0 1/20 0.30
FYN P06241 1/20 0.30
GRIN1 Q05586 1/20 0.30
GRIN2A Q12879 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23215199 0.73 EGLN2 (0.47) EGLN2
SCHEMBL12646055 0.66 HTR2A (0.40) KMT2AALDH1A1THRBHPGD
SCHEMBL13209735 0.65 HPGD (0.41) KMT2AALDH1A1KDM4EPOLBHPGD
SCHEMBL1691581 0.61 MKNK1 (0.47) ALDH1A1HPGDFYN
SCHEMBL13024178 0.60 IDH1 (0.62) KMT2AALDH1A1THRBKDM4EHPGD
SCHEMBL13024189 0.59 HDAC4 (0.70) KMT2AALDH1A1THRBMAPT
SCHEMBL18078708 0.59 ALDH1A1 (0.42) KMT2AALDH1A1KDM4EHPGDGLA
SCHEMBL8378548 0.59 FYN (0.35) KMT2AALDH1A1KDM4EHPGDTP53
SCHEMBL26538138 0.58 BAZ2B (0.41) KMT2ATHRBKDM4EPOLBMAPT
SCHEMBL19491595 0.58

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5019578-A β-adrenergic agonists MERCK & CO., INC. (US) 1991-05-28 US disclosed
EP-0318092-A2 Novel beta-adrenergic agonists MERCK & CO. INC. (US) 1989-05-31 EP disclosed