SCHEMBL9770286

SCHEMBL9770286

CSC(N)c1ccc(O)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 8/20 0.48
ESR2 Q92731 7/20 0.48
PDCD1 Q15116 1/20 0.48
CD274 Q9NZQ7 1/20 0.48
ALOX15 P16050 3/20 0.43
TDP1 Q9NUW8 3/20 0.43
SLC6A2 P23975 2/20 0.43
LMNA P02545 2/20 0.43
CYP3A4 P08684 2/20 0.43
MAPT P10636 2/20 0.43
CYP2C9 P11712 2/20 0.43
CYP1A2 P05177 1/20 0.43
PGR P06401 1/20 0.43
CHRM2 P08172 1/20 0.43
ADORA3 P0DMS8 1/20 0.43
AR P10275 1/20 0.43
CYP2D6 P10635 1/20 0.43
CHRM1 P11229 1/20 0.43
DRD1 P21728 1/20 0.43
TBXA2R P21731 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL109302 0.75 DPP4 (0.50) LMNATAAR1HIF1AKDM4EALDH1A1
SCHEMBL9522260 0.74 ADRB1 (0.56) ESR1ESR2TDP1LMNACYP3A4
Hydrochloric Acid SCHEMBL10435080 0.73 DPP4 (0.48) LMNATAAR1HIF1AKDM4EALDH1A1
SCHEMBL19304127 0.73 ESR1 (0.56) ESR1ESR2PDCD1CD274ALOX15
SCHEMBL24369694 0.73 CYP1A2 (0.50) TDP1CYP3A4CYP1A2CYP2D6CYP2C19
SCHEMBL2032476 0.72 ESR1 (0.62) ESR1ESR2PDCD1CD274ALOX15
SCHEMBL633374 0.72 ESR1 (0.62) ESR1ESR2PDCD1CD274ALOX15
SCHEMBL2037513 0.72 ESR1 (0.62) ESR1ESR2PDCD1CD274ALOX15
SCHEMBL24897061 0.71 CYP2A6 (0.43) CYP3A4CYP2C19TSHRALDH1A1CA12
SCHEMBL8607150 0.71 ESR1 (0.52) ESR1ESR2PDCD1CD274ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017156179-A1 3-PHOSPHOGLYCERATE DEHYDROGENASE INHIBITORS AND USES THEREOF RAZE THERAPEUTICS, INC. (US) 2017-09-14 WO disclosed
US-5053053-A PROCESS FOR DYEING KERATINOUS FIBRES WITH A HYDROXYINDOLE IN COMBINATION WITH A QUINONE DERIVATIVE; AND NOVEL 1,4-BENZOQUINONES L'OREAL (FR) 1991-10-01 US disclosed