SCHEMBL9771971

SCHEMBL9771971

CN1CCc2cc(Cl)c(OC(=O)NC3CCCCC3)cc2C(c2ccc3cccoc2-3)C1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD1 P21728 11/20 0.44
DRD5 P21918 6/20 0.39
DRD2 P14416 4/20 0.39
KDM4E B2RXH2 1/20 0.39
ALPL P05186 1/20 0.39
ALPI P09923 1/20 0.39
GAA P10253 1/20 0.39
ALPG P10696 1/20 0.39
CYP1A2 P05177 2/20 0.37
CYP2D6 P10635 2/20 0.37
TSHR P16473 2/20 0.37
HSD17B10 Q99714 2/20 0.37
CYP3A4 P08684 1/20 0.37
NFKB1 P19838 1/20 0.37
THPO P40225 1/20 0.37
MEN1 O00255 1/20 0.37
ALOX15 P16050 1/20 0.37
KMT2A Q03164 1/20 0.37
SIGMAR1 Q99720 1/20 0.37
FAAH O00519 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9529171 0.88 DRD1 (0.45) DRD1DRD5DRD2CYP1A2CYP2D6
SCHEMBL9771968 0.86 DRD1 (0.62) DRD1DRD5DRD2KDM4EALPL
SCHEMBL9529550 0.85 DRD1 (0.47) DRD1DRD5DRD2CYP1A2CYP2D6
SCHEMBL9529141 0.84 DRD1 (0.43) DRD1DRD5DRD2CYP1A2CYP2D6
SCHEMBL9530502 0.84 DRD1 (0.45) DRD1DRD5DRD2CYP1A2CYP2D6
SCHEMBL9528456 0.84 DRD1 (0.43) DRD1DRD5DRD2CYP1A2CYP2D6
SCHEMBL9772051 0.84 DRD1 (0.44) DRD1DRD5DRD2CYP1A2CYP2D6
SCHEMBL10691057 0.81 DRD1 (0.53) DRD1DRD5DRD2CYP1A2CYP2D6
SCHEMBL9771938 0.81 DRD1 (0.41) DRD1DRD5DRD2CYP1A2CYP2D6
SCHEMBL9528077 0.80 DRD1 (0.40) DRD1DRD5DRD2CYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5017571-A Prodrugs, mental disorders NOVO NORDISK A/S (DK) 1991-05-21 US disclosed
EP-0331130-A1 Carbamic acid ester of substituted 7-hydroxy-2,3,4,5-tetrahydro-1H-3-benzazepines NOVO NORDISK A/S (DK) 1989-09-06 EP disclosed