SCHEMBL9778530

SCHEMBL9778530

COc1ccc(C2SCCCS2)cc1OCc1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 1/20 0.55
PDE4B Q07343 1/20 0.55
PDE4C Q08493 1/20 0.55
PDE4D Q08499 1/20 0.55
TSHR P16473 1/20 0.51
APP P05067 2/20 0.47
MAPK1 P28482 1/20 0.47
HSD17B10 Q99714 1/20 0.47
SMPD1 P17405 1/20 0.46
HDAC1 Q13547 1/20 0.46
HDAC8 Q9BY41 1/20 0.46
HDAC6 Q9UBN7 1/20 0.46
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
CSF1R P07333 1/20 0.44
SIRT2 Q8IXJ6 1/20 0.44
PRMT5 O14744 1/20 0.43
KMT2A Q03164 2/20 0.43
MEN1 O00255 1/20 0.43
LMNA P02545 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9778660 0.95 APP (0.53) PDE4APDE4BPDE4CPDE4DTSHR
SCHEMBL9778946 0.95 PDE4A (0.57) PDE4APDE4BPDE4CPDE4DTSHR
SCHEMBL9778560 0.92 PDE4A (0.44) PDE4APDE4BPDE4CPDE4DTSHR
SCHEMBL9778888 0.90 APP (0.55) PDE4APDE4BPDE4CPDE4DTSHR
SCHEMBL9778863 0.89 KDM4E (0.47) PDE4APDE4BPDE4CPDE4DTSHR
SCHEMBL9778588 0.86 PDE4A (0.46) PDE4APDE4BPDE4CPDE4DAPP
SCHEMBL9778549 0.84 PDE4A (0.54) PDE4APDE4BPDE4CPDE4DAPP
SCHEMBL9778662 0.83 MAPT (0.48) PDE4APDE4BPDE4CPDE4DAPP
SCHEMBL9778679 0.82 HIF1A (0.49) TSHR
SCHEMBL9778850 0.82 TSHR (0.57) PDE4APDE4BPDE4CPDE4DTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5063197-A Aromatic compound MITSUBISHI PAPER MILLS LIMITED (JP) 1991-11-05 US disclosed
US-4127588-A Sulphur containing derivatives HOFFMANN-LA ROCHE INC. (US) 1978-11-28 US disclosed
US-4073797-A CORONARY DILATOR HOFFMANN-LA ROCHE INC. (US) 1978-02-14 US disclosed
US-4003914-A DITHIANE AND DISULFONE CORONARY DILATING AGENTS HOFFMANN-LA ROCHE INC. (US) 1977-01-18 US disclosed