SCHEMBL9779057

SCHEMBL9779057

Cn1cc(C=O)c2ccc3cc4ccccc4cc3c21

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.49
IMPDH2 P12268 1/20 0.49
KDM4E B2RXH2 1/20 0.41
ERN1 O75460 3/20 0.36
CYP2A6 P11509 2/20 0.36
CYP1A2 P05177 1/20 0.36
TDP1 Q9NUW8 1/20 0.35
PIM1 P11309 4/20 0.35
PIM3 Q86V86 4/20 0.35
PIM2 Q9P1W9 1/20 0.35
POLB P06746 3/20 0.34
L3MBTL1 Q9Y468 1/20 0.33
MEN1 O00255 1/20 0.33
PTPN1 P18031 1/20 0.33
KMT2A Q03164 1/20 0.33
NPC1 O15118 1/20 0.33
LMNA P02545 1/20 0.33
MAPT P10636 1/20 0.33
HPGD P15428 1/20 0.33
HTT P42858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9779010 0.83 ALDH1A1 (0.54) ALDH1A1IMPDH2KDM4EERN1CYP2A6
SCHEMBL5440842 0.74 KDM4E (0.43) ALDH1A1IMPDH2KDM4EERN1TDP1
SCHEMBL14156855 0.72 ALDH1A1 (0.59) ALDH1A1IMPDH2KDM4ETDP1PIM1
SCHEMBL1093997 0.69 ALDH1A1 (0.56) ALDH1A1IMPDH2KDM4ECYP2A6CYP1A2
SCHEMBL29392367 0.69 ALDH1A1 (0.50) ALDH1A1KDM4EERN1CYP2A6CYP1A2
SCHEMBL39718 0.69 ALDH1A1 (0.50) ALDH1A1KDM4EERN1CYP2A6CYP1A2
SCHEMBL347177 0.68 ERN1 (0.43) ALDH1A1KDM4EERN1CYP2A6CYP1A2
Methyl Alcohol SCHEMBL27597852 0.68 ALDH1A1 (0.46) ALDH1A1KDM4EERN1CYP2A6CYP1A2
SCHEMBL838056 0.68 ALDH1A1 (0.54) ALDH1A1IMPDH2KDM4ECYP2A6CYP1A2
SCHEMBL1093392 0.68 ALDH1A1 (0.54) ALDH1A1IMPDH2KDM4EERN1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4999369-A Antitumor agents BURROUGHS WELLCOME CO. (US) 1991-03-12 US disclosed
EP-0246077-B1 HETEROPOLYCYCLIC AROMATIC COMPOUNDS THE WELLCOME FOUNDATION LIMITED (GB) 1990-11-22 EP disclosed
US-4910218-A With a hydroxy containing secondary amine group BURROUGHS WELLCOME CO. (US) 1990-03-20 US disclosed
EP-0246077-A1 Heteropolycyclic aromatic compounds THE WELLCOME FOUNDATION LIMITED (GB) 1987-11-19 EP disclosed