SCHEMBL9780487

SCHEMBL9780487

CCCc1c(OCCCSc2ccc(CC(O)C(C)C(=O)OC)cc2)ccc(C(C)=O)c1O

nearest known ligand 0.62

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYSLTR2 Q9NS75 11/20 0.62
CYSLTR1 Q9Y271 11/20 0.62
PPARG P37231 4/20 0.53
PPARD Q03181 4/20 0.53
PPARA Q07869 4/20 0.53
GRM2 Q14416 2/20 0.47
LMNA P02545 1/20 0.47
CYP1A2 P05177 1/20 0.47
MAPT P10636 1/20 0.47
CYP2C9 P11712 1/20 0.47
NFKB1 P19838 1/20 0.47
BLM P54132 1/20 0.47
PDE5A O76074 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9735067 0.91 CYSLTR2 (0.67) CYSLTR2CYSLTR1PPARGPPARDPPARA
SCHEMBL10915351 0.89 CYSLTR2 (0.57) CYSLTR2CYSLTR1PPARGPPARDPPARA
SCHEMBL9780267 0.88 CYSLTR2 (0.57) CYSLTR2CYSLTR1PPARGPPARDPPARA
SCHEMBL9780317 0.86 CYSLTR2 (0.55) CYSLTR2CYSLTR1PPARGPPARDPPARA
SCHEMBL10893732 0.84 CYSLTR2 (0.61) CYSLTR2CYSLTR1PPARGPPARDPPARA
SCHEMBL6137114 0.82 PPARG (0.75) CYSLTR2CYSLTR1PPARGPPARDPPARA
SCHEMBL9734508 0.82 CYSLTR2 (0.59) CYSLTR2CYSLTR1PPARGPPARDPPARA
SCHEMBL9780216 0.81 CYSLTR2 (0.49) CYSLTR2CYSLTR1PPARGPPARDPPARA
SCHEMBL9734155 0.79 PPARG (0.67) CYSLTR2CYSLTR1PPARGPPARDPPARA
SCHEMBL9780479 0.79 CYSLTR2 (0.84) CYSLTR2CYSLTR1PPARGPPARDPPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0206741-B1 LEUKOTRIENE ANTAGONISTS MERCK FROSST CANADA INC. (CA) 1991-04-10 EP disclosed
US-4990526-A Skin disorders, antiallergens, antiinflammatory agents MERCK FROSST CANADA, INC. (CA) 1991-02-05 US disclosed