SCHEMBL9780678

SCHEMBL9780678

CC(Cc1c(Cl)cccc1Cl)C(=O)O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 1/20 0.52
POLB P06746 2/20 0.44
ALDH1A1 P00352 2/20 0.44
HPGD P15428 2/20 0.44
KMT2A Q03164 4/20 0.42
APAF1 O14727 2/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
KDM4E B2RXH2 2/20 0.41
MAPT P10636 1/20 0.41
RECQL P46063 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
CXCL8 P10145 1/20 0.41
HTT P42858 1/20 0.40
TBXAS1 P24557 1/20 0.40
MEN1 O00255 1/20 0.40
LMNA P02545 1/20 0.40
CYP3A4 P08684 1/20 0.40
HTR1A P08908 1/20 0.40
ADRA2A P08913 1/20 0.40
CYP2D6 P10635 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9780682 1.00 AKR1B1 (0.52) AKR1B1POLBALDH1A1HPGDKMT2A
SCHEMBL13235859 0.85 AKR1B1 (0.47) AKR1B1POLBALDH1A1HPGDKMT2A
SCHEMBL14208222 0.79 PPARG (0.53) POLBALDH1A1APAF1L3MBTL1KDM4E
SCHEMBL1454266 0.79 PPARG (0.53) POLBALDH1A1APAF1L3MBTL1KDM4E
SCHEMBL27943299 0.79 AKR1B1 (0.46) AKR1B1POLBALDH1A1HPGDKMT2A
SCHEMBL9780828 0.79 KMT2A (0.49) AKR1B1POLBALDH1A1HPGDKMT2A
SCHEMBL9780837 0.79 KMT2A (0.49) AKR1B1POLBALDH1A1HPGDKMT2A
SCHEMBL11863668 0.78 AKR1B1 (0.59) AKR1B1POLBALDH1A1HPGDKMT2A
SCHEMBL7136191 0.77 APAF1 (0.41) POLBALDH1A1HPGDAPAF1L3MBTL1
SCHEMBL29397997 0.77 SLC7A5 (0.55) AKR1B1KMT2AMEN1CYP2C19HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0257378-B1 PYRIMIDINE DERIVATIVES, THEIR PREPARATION AND MEDICAMENTS CONTAINING THESE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1991-07-03 EP disclosed
US-5010060-A Method of treating herpes simplex viral infection employing pyrimidine derivatives HOFFMANN-LA ROCHE INC. (US) 1991-04-23 US disclosed
US-4851519-A AMIDO NUCLEOSIDES, VIRICIDES HOFFMANN-LA ROCHE INC. (US) 1989-07-25 US disclosed
EP-0257378-A1 Pyrimidine derivatives, their preparation and medicaments containing these derivatives F. HOFFMANN-LA ROCHE AG (CH) 1988-03-02 EP disclosed