SCHEMBL9782425

SCHEMBL9782425

CC(O)[C@H]1C(=O)N2C(C(=O)OCc3ccccc3)=CC[C@@H]12

nearest known ligand 0.52

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ELANE P08246 14/20 0.52
GPBAR1 Q8TDU6 1/20 0.42
SLC6A2 P23975 1/20 0.40
SLC6A3 Q01959 1/20 0.40
KMT2A Q03164 1/20 0.40
TDP1 Q9NUW8 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11061309 1.00 ELANE (0.52) ELANEGPBAR1SLC6A2SLC6A3KMT2A
SCHEMBL9782863 0.92 ELANE (0.55) ELANEGPBAR1SLC6A2SLC6A3KMT2A
SCHEMBL11486285 0.88 ELANE (0.47) ELANEGPBAR1
SCHEMBL11062621 0.88 ELANE (0.43) ELANEGPBAR1SLC6A2SLC6A3KMT2A
SCHEMBL11061674 0.84 ELANE (0.43) ELANEGPBAR1SLC6A2SLC6A3KMT2A
SCHEMBL11063454 0.83 ELANE (0.45) ELANESLC6A2SLC6A3KMT2ATDP1
SCHEMBL9698851 0.81 ELANE (0.34) ELANESLC6A2TDP1
SCHEMBL11063535 0.80 FOLH1 (0.43) ELANESLC6A2SLC6A3KMT2ATDP1
SCHEMBL11276416 0.80 ELANE (0.55) ELANEGPBAR1
SCHEMBL11061653 0.80 ELANE (0.42) ELANESLC6A2SLC6A3KMT2ATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5055573-A Reacting substituted azetidinone with glyoxalate ester, halogenating, reacting with phosphine, oxidizing, cyclizing, deprotecting MERCK & CO., INC. (US) 1991-10-08 US disclosed
US-4775669-A ANTIBIOTIC MERCK & CO., INC. (US) 1988-10-04 US disclosed
US-4543257-A PENICILLIN ANTIBIOTICS MERCK & CO., INC. (US) 1985-09-24 US disclosed
US-4348320-A PENICILLIN INTERMEDIATES MERCK & CO., INC. (US) 1982-09-07 US disclosed