SCHEMBL9788780

SCHEMBL9788780

O=C(CCc1cccc(F)c1)c1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.54
RAB9A P51151 2/20 0.54
CASP3 P42574 2/20 0.54
TDP1 Q9NUW8 2/20 0.54
SENP8 Q96LD8 1/20 0.54
SENP7 Q9BQF6 1/20 0.54
SENP6 Q9GZR1 1/20 0.54
GPR52 Q9Y2T5 1/20 0.51
HSD11B1 P28845 1/20 0.50
FFAR1 O14842 1/20 0.50
NR4A2 P43354 3/20 0.49
TAAR1 Q96RJ0 1/20 0.49
CASP7 P55210 1/20 0.48
ALDH1A1 P00352 1/20 0.47
GAA P10253 1/20 0.47
CYP2C19 P33261 1/20 0.47
L3MBTL1 Q9Y468 2/20 0.47
LMNA P02545 1/20 0.47
MAPT P10636 1/20 0.47
CES2 O00748 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29580879 1.00 NPC1 (0.54) NPC1RAB9ACASP3TDP1SENP8
SCHEMBL28128458 0.90 GPR52 (0.58) NPC1RAB9ACASP3TDP1SENP8
SCHEMBL29579853 0.90 GPR52 (0.58) NPC1RAB9ACASP3TDP1SENP8
SCHEMBL11443407 0.87 DPP4 (0.53) NPC1RAB9ACASP3TDP1FFAR1
SCHEMBL570730 0.83 MAPT (0.51) NPC1RAB9AGPR52NR4A2L3MBTL1
SCHEMBL334758 0.82 FFAR1 (0.68) CASP3FFAR1TAAR1CASP7
SCHEMBL30572 0.82 TDP1 (0.77) NPC1RAB9ACASP3TDP1SENP8
SCHEMBL15524969 0.82 TDP1 (0.77) NPC1RAB9ACASP3TDP1SENP8
SCHEMBL28251466 0.82 TDP1 (0.77) NPC1RAB9ACASP3TDP1SENP8
SCHEMBL8008357 0.81 NPC1 (0.56) NPC1RAB9ACASP3TDP1SENP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111499503-B Method for synthesizing alpha-alkylated ketone in water 南京理工大学 2022-04-08 CN disclosed
CN-114288294-A Compounds and methods for treating or preventing hematologic cancers 布罗德研究所股份有限公司 2022-04-08 CN disclosed
CN-111499503-A Method for synthesizing α -alkylated ketone in water 南京理工大学 2020-08-07 CN disclosed
US-5032597-A Antitumor DU PONT MERCK PHARMACEUTICAL (US) 1991-07-16 US disclosed
EP-0133244-B1 PHENYLQUINOLINECARBOXYLIC ACIDS AND DERIVATIVES AS ANTITUMOR AGENTS E.I. DU PONT DE NEMOURS AND COMPANY (US) 1990-12-05 EP disclosed
EP-0133244-A2 Phenylquinolinecarboxylic acids and derivatives as antitumor agents E.I. DU PONT DE NEMOURS AND COMPANY (US) 1985-02-20 EP disclosed