SCHEMBL9795384

SCHEMBL9795384

CC(C(=O)c1ccc(C(F)(F)F)cn1)n1cncn1

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.47
SCN9A Q15858 1/20 0.38
MAPT P10636 1/20 0.38
HSP90AA1 P07900 1/20 0.38
HDAC1 Q13547 1/20 0.37
HDAC8 Q9BY41 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
EPHX2 P34913 1/20 0.36
POLB P06746 1/20 0.36
CYP3A4 P08684 1/20 0.36
L3MBTL1 Q9Y468 3/20 0.36
KDM4E B2RXH2 2/20 0.36
PDE4D Q08499 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
MAPK1 P28482 1/20 0.36
HRH3 Q9Y5N1 2/20 0.35
ACACB O00763 1/20 0.35
ABL1 P00519 1/20 0.35
LMNA P02545 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10361626 0.82 HSP90AA1 (0.49) KMT2AMAPTHSP90AA1HDAC1HDAC8
SCHEMBL9792762 0.81 CYP3A4 (0.46) KMT2AMAPTHSP90AA1POLBCYP3A4
Nitric Acid SCHEMBL9795438 0.79 KMT2A (0.34) KMT2AMAPTHSP90AA1HDAC1HDAC8
SCHEMBL18358401 0.76 KMT2A (0.62) KMT2ASCN9AMAPTPOLBKDM4E
Nitric Acid SCHEMBL9795407 0.75 CYP19A1 (0.37) KMT2ASCN9AMAPTPOLBCYP3A4
SCHEMBL9795320 0.74 KMT2A (0.58) KMT2ASCN9AMAPTPOLBKDM4E
SCHEMBL9388155 0.73 MAPT (0.44) KMT2AMAPTHSP90AA1HDAC1HDAC8
Nitric Acid SCHEMBL10587061 0.73 KMT2A (0.35) KMT2ASCN9AMAPTHSP90AA1KDM4E
SCHEMBL27244049 0.72 KMT2A (0.64) KMT2ASCN9APOLBKDM4ESMN1; SMN2
SCHEMBL10709771 0.70 MAPT (0.43) KMT2AMAPTHSP90AA1HDAC1HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5032607-A Enzyme inhibitors IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1991-07-16 US disclosed
US-4866086-A PHENYLTRIAZOLYL OLEFINIC AROMATASE INHIBITORS IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1989-09-12 US disclosed
EP-0299683-A2 Heterocyclic olefinic compounds and their use as aromatase inhibitors IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1989-01-18 EP disclosed