SCHEMBL9796281

SCHEMBL9796281

CC(C)S(=O)(=O)Oc1cn(C)c2cc(F)ccc2c1=O

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.42
GSK3B P49841 3/20 0.36
PRKCA P17252 1/20 0.36
IDO1 P14902 1/20 0.36
TDO2 P48775 1/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
SCN9A Q15858 2/20 0.36
BRD4 O60885 4/20 0.35
CNR2 P34972 2/20 0.35
DRD2 P14416 1/20 0.35
SLC6A4 P31645 1/20 0.35
PER2 O15055 1/20 0.34
CRY1 Q16526 1/20 0.34
CRY2 Q49AN0 1/20 0.34
TP53 P04637 1/20 0.34
HTR6 P50406 2/20 0.33
CNR1 P21554 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9796452 0.85 ATM (0.44) ATMGSK3BPRKCAIDO1TDO2
SCHEMBL9796420 0.83 ATM (0.43) ATMGSK3BPRKCAIDO1TDO2
SCHEMBL9796513 0.75 ALDH1A1 (0.48) GSK3BKDM4EALDH1A1BRD4DRD2
SCHEMBL6050597 0.72 ATM (0.48) ATMIDO1TDO2KDM4EALDH1A1
SCHEMBL5441907 0.72 ATM (0.44) ATMIDO1TDO2KDM4EALDH1A1
SCHEMBL9796456 0.72 ATM (0.42) ATMGSK3BPRKCAIDO1TDO2
SCHEMBL10629394 0.71 ATM (0.47) ATMIDO1TDO2KDM4EALDH1A1
SCHEMBL9796325 0.70 TP53 (0.41) GSK3BPRKCAKDM4EALDH1A1SCN9A
SCHEMBL1606274 0.70 IDO1 (0.43) ATMGSK3BPRKCAIDO1TDO2
SCHEMBL9796252 0.70 ATM (0.51) ATMGSK3BPRKCAIDO1TDO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4997840-A Quinolone sulphonates having antihypertensive activity THE BOOTS COMPANY, PLC (GB) 1991-03-05 US disclosed
EP-0330340-A1 Therapeutic agents The Boots Company PLC (GB) 1989-08-30 EP disclosed
WO-1989007593-A1 THERAPEUTIC AGENTS THE BOOTS COMPANY PLC (GB) 1989-08-24 WO disclosed