SCHEMBL9804079

SCHEMBL9804079

O=C(C=Cc1ccc(Cl)cc1)c1cccnc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAPT P10636 6/20 1.00
CYP1A1 P04798 7/20 0.75
CYP1A2 P05177 7/20 0.75
CYP1B1 Q16678 7/20 0.75
CYP3A4 P08684 5/20 0.75
CYP2D6 P10635 5/20 0.75
ALDH1A1 P00352 4/20 0.68
KMT2A Q03164 2/20 0.68
MEN1 O00255 1/20 0.68
LMNA P02545 4/20 0.67
MAOB P27338 1/20 0.67
KDM4E B2RXH2 1/20 0.67
PKM P14618 1/20 0.67
APP P05067 1/20 0.66
GSK3B P49841 1/20 0.66
MAPK1 P28482 1/20 0.64
NPSR1 Q6W5P4 1/20 0.64
HPGD P15428 1/20 0.63
HSP90AA1 P07900 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2705060 1.00 MAPT (1.00) MAPTCYP1A1CYP1A2CYP1B1CYP3A4
SCHEMBL1604142 0.86 CYP1A1 (0.77) MAPTCYP1A1CYP1A2CYP1B1CYP3A4
SCHEMBL31436361 0.86 CYP1A1 (0.77) MAPTCYP1A1CYP1A2CYP1B1CYP3A4
SCHEMBL1322027 0.86 CYP1A1 (0.82) MAPTCYP1A1CYP1A2CYP1B1CYP3A4
SCHEMBL31436369 0.86 CYP1A1 (0.77) MAPTCYP1A1CYP1A2CYP1B1CYP3A4
SCHEMBL1322029 0.86 CYP1A1 (0.82) MAPTCYP1A1CYP1A2CYP1B1CYP3A4
SCHEMBL979408 0.86 CYP1B1 (1.00) MAPTCYP1A1CYP1A2CYP1B1CYP3A4
SCHEMBL20570877 0.86 CYP1A1 (0.82) MAPTCYP1A1CYP1A2CYP1B1CYP3A4
SCHEMBL9503680 0.86 CYP1B1 (1.00) MAPTCYP1A1CYP1A2CYP1B1CYP3A4
SCHEMBL3024151 0.85 CYP1B1 (0.75) MAPTCYP1A1CYP1A2CYP1B1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2167058-B1 FAMILY OF PFKFB3 INHIBITORS WITH ANTI-NEOPLASTIC ACTIVITIES UNIV LOUISVILLE RES FOUND (US) 2015-08-12 EP disclosed
EP-0214566-B1 3-PROPENYL PYRIDINES AND THEIR USE AS FUNGICIDES BASF Aktiengesellschaft (DE) 1991-03-13 EP disclosed
EP-0214566-A2 3-Propenyl pyridines and their use as fungicides BASF Aktiengesellschaft (DE) 1987-03-18 EP disclosed