SCHEMBL9804830

SCHEMBL9804830

N#CC(CCc1ccc(Cl)cc1)(Cc1cncnc1)c1cccc(C(F)(F)F)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 6/20 0.39
CTSC P53634 2/20 0.37
MAPT P10636 2/20 0.35
HTT P42858 2/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
VNN1 O95497 2/20 0.35
TP53 P04637 1/20 0.34
POLB P06746 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
P2RX3 P56373 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
CNR1 P21554 1/20 0.34
GRIN1 Q05586 1/20 0.34
GRIN2B Q13224 1/20 0.34
KCNH2 Q12809 1/20 0.33
CHIT1 Q13231 1/20 0.33
CHIA Q9BZP6 1/20 0.33
ALDH1A1 P00352 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9804733 0.89 CYP19A1 (0.47) CYP19A1
SCHEMBL9804866 0.86 CYP19A1 (0.45) CYP19A1ALDH1A1
SCHEMBL9804735 0.85 CYP19A1 (0.42) CYP19A1CTSCMAPTHTTMEN1
SCHEMBL9804822 0.85 CYP19A1 (0.42) CYP19A1ALDH1A1
SCHEMBL9804762 0.82 CTSC (0.39) CYP19A1CTSCMEN1KMT2AVNN1
SCHEMBL9804745 0.79 CYP19A1 (0.44) CYP19A1CNR1ALDH1A1
SCHEMBL9804836 0.77 EBP (0.41) CYP19A1ALDH1A1HPGD
SCHEMBL9804729 0.76 CYP19A1 (0.52) CYP19A1
SCHEMBL10371112 0.75 CYP3A4 (0.46) CYP19A1MAPT
SCHEMBL10371526 0.75 CYP19A1 (0.46) CYP19A1CTSCHTTNPSR1VNN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0276920-B1 (2-CYANO-2-(PHENYL OR NAPHTHYL)-2-SUBSTITUTED-ETHYL) PYRAZINES, PYRIMIDINES AND PYRIDAZINES ROHM AND HAAS COMPANY (US) 1991-04-03 EP disclosed
EP-0276920-A1 (2-Cyano-2-(phenyl or naphthyl)-2-substituted-ethyl) pyrazines, pyrimidines and pyridazines ROHM AND HAAS COMPANY (US) 1988-08-03 EP disclosed