SCHEMBL9804745

SCHEMBL9804745

N#CC(CCc1ccc(Cl)cc1)(Cc1cncnc1)c1ccccc1Cl

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 8/20 0.44
CYP3A4 P08684 2/20 0.34
CYP3A5 P20815 1/20 0.34
CNR1 P21554 1/20 0.34
CNR2 P34972 1/20 0.34
ALDH1A1 P00352 1/20 0.32
CTSL P07711 1/20 0.32
CTSS P25774 1/20 0.32
CTSK P43235 1/20 0.32
NR1D1 P20393 1/20 0.32
NR1H3 Q13133 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9804866 0.88 CYP19A1 (0.45) CYP19A1CYP3A4CYP3A5ALDH1A1CTSL
SCHEMBL9804822 0.86 CYP19A1 (0.42) CYP19A1CYP3A4CYP3A5ALDH1A1CTSL
SCHEMBL9804841 0.84 CYP3A4 (0.38) CYP19A1CYP3A4CYP3A5ALDH1A1NR1D1
SCHEMBL9804762 0.81 CTSC (0.39) CYP19A1CNR1
SCHEMBL9557095 0.79 ALDH1A1 (0.53) CYP19A1CYP3A4ALDH1A1
SCHEMBL9804733 0.79 CYP19A1 (0.47) CYP19A1CYP3A4CYP3A5
SCHEMBL9804830 0.79 CYP19A1 (0.39) CYP19A1CNR1ALDH1A1
SCHEMBL9804729 0.79 CYP19A1 (0.52) CYP19A1CYP3A4CYP3A5
SCHEMBL9804836 0.78 EBP (0.41) CYP19A1CYP3A4ALDH1A1CTSL
SCHEMBL9804674 0.77 CYP19A1 (0.49) CYP19A1CYP3A4CYP3A5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0276920-B1 (2-CYANO-2-(PHENYL OR NAPHTHYL)-2-SUBSTITUTED-ETHYL) PYRAZINES, PYRIMIDINES AND PYRIDAZINES ROHM AND HAAS COMPANY (US) 1991-04-03 EP disclosed
EP-0276920-A1 (2-Cyano-2-(phenyl or naphthyl)-2-substituted-ethyl) pyrazines, pyrimidines and pyridazines ROHM AND HAAS COMPANY (US) 1988-08-03 EP disclosed